A High-Throughput Screening Compatible Assay for Activators and Inhibitors of Methionine Sulfoxide Reductase A

door Brunell, David, Weissbach, Herbert, Hodder, Peter, Brot, Nathan
Gepubliceerd in 2010

Monitoring of HTS Compound Library Quality via a High-Resolution Image Acquisition and Processing Instrument

door Baillargeon, Pierre, Scampavia, Louis, Einsteder, Ross, Hodder, Peter
Gepubliceerd in 2011

Synthesis of Small Molecule Inhibitors of the Orphan Nuclear Receptor Steroidogenic Factor-1 (NR5A1) Based on Isoquinolinone Scaffolds

door Roth, Joshua, Madoux, Franck, Hodder, Peter, Roush, William R.
Gepubliceerd in 2008

Inhibition of Adrenocortical Carcinoma Cell Proliferation by Steroidogenic Factor-1 Inverse Agonists

door Doghman, Mabrouka, Cazareth, Julie, Douguet, Dominique, Madoux, Franck, Hodder, Peter, Lalli, Enzo
Gepubliceerd in 2009

Dynamics of the formation of a hydrogel by a pathogenic amyloid peptide: islet amyloid polypeptide

door Jean, Létitia, Lee, Chiu Fan, Hodder, Peter, Hawkins, Nick, Vaux, David J.
Gepubliceerd in Sci Rep (2016)

Inhibition of Adrenocortical Carcinoma Cell Proliferation by Steroidogenic Factor-1 Inverse Agonists

door Doghman, Mabrouka, Cazareth, Julie, Douguet, Dominique, Madoux, Franck, Hodder, Peter, Lalli, Enzo
Gepubliceerd in Mol Endocrinol (2009)

An altered zinc-binding site confers resistance to a covalent inactivator of New Delhi metallo-beta-lactamase-1 (NDM-1) discovered by high-throughput screening

door Thomas, Pei W., Spicer, Timothy, Cammarata, Michael, Brodbelt, Jennifer S., Hodder, Peter, Fast, Walter
Gepubliceerd in 2013

High Throughput Screen for Pharmacoperones of the Vasopressin Type 2 Receptor

door Conn, P. Michael, Smith, Emery, Hodder, Peter, Janovick, Jo Ann, Smithson, David C.
Gepubliceerd in 2013

Development of an HTS-Compatible Assay for the Discovery of ASK1 Signalosome Inhibitors Using AlphaScreen Technology

door Sturchler, Emmanuel, Chen, Weimin, Spicer, Timothy, Hodder, Peter, McDonald, Patricia, Duckett, Derek
Gepubliceerd in 2014

In Pursuit of Synthetic Modulators for the Orphan Retina-Specific Nuclear Receptor NR2E3

door Qin, Qiong, Knapinska, Anna, Dobri, Nicoleta, Madoux, Franck, Chase, Peter, Hodder, Peter, Petrukhin, Konstantin
Gepubliceerd in 2013

An Ultra-High Throughput Cell-Based Screen for Wee1 Degradation Inhibitors

door MADOUX, FRANCK, SIMANSKI, SCOTT, CHASE, PETER, MISHRA, JITENDRA K., ROUSH, WILLIAM R., AYAD, NAGI G., HODDER, PETER
Gepubliceerd in 2010

Identification of Novel, Exosite-Binding Matrix Metalloproteinase-13 Inhibitor Scaffolds

door Roth, Joshua, Minond, Dmitriy, Darout, Etzer, Liu, Qin, Lauer, Janelle, Hodder, Peter, Fields, Gregg B., Roush, William R.
Gepubliceerd in 2011

A FluoPol-ABPP PAD2 High-Throughput Screen Identifies the First Calcium Site Inhibitor Targeting the PADs

door Lewallen, Daniel M., Bicker, Kevin L., Madoux, Franck, Chase, Peter, Anguish, Lynne, Coonrod, Scott, Hodder, Peter, Thompson, Paul R.
Gepubliceerd in 2014

High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate

door Lauer-Fields, Janelle L., Minond, Dmitriy, Chase, Peter S., Baillargeon, Pierre E., Saldanha, S. Adrian, Stawikowska, Roma, Hodder, Peter, Fields, Gregg B.
Gepubliceerd in 2008

Screening of potential ADAMTS-4 inhibitors utilizing a collagen-model FRET substrate

door Lauer-Fields, Janelle L., Spicer, Timothy P., Chase, Peter S., Cudic, Mare, Burstein, Gayle D., Nagase, Hideaki, Hodder, Peter, Fields, Gregg B.
Gepubliceerd in 2007

Discovery, synthesis and SAR analysis of novel selective small molecule S1P(4)–R agonists based on a (2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-one chem...

door Urbano, Mariangela, Guerrero, Miguel, Velaparthi, Subash, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
Gepubliceerd in 2011

Potent and Selective Inhibitors of Glutathione S-transferase Omega 1 that Impair Cancer Drug Resistance

door Tsuboi, Katsunori, Bachovchin, Daniel A., Speers, Anna E., Spicer, Timothy P., Fernandez-Vega, Virneliz, Hodder, Peter, Rosen, Hugh, Cravatt, Benjamin F.
Gepubliceerd in 2011

Potent, selective and cell penetrant inhibitors of SF-1 by functional uHTS

door Madoux, Franck, Li, Xiaolin, Chase, Peter, Zastrow, Gina, Cameron, Michael D., Conkright, Juliana J., Griffin, Patrick R., Thacher, Scott, Hodder, Peter
Gepubliceerd in 2008

Discovery, Design and Synthesis of Novel Potent and Selective Sphingosine-1-Phosphate 4 Receptor (S1P(4)-R) Agonists

door Guerrero, Miguel, Urbano, Mariangela, Zhao, Jian, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
Gepubliceerd in 2011

Inhibiting AMPylation: A novel screen to identify the first small molecule inhibitors of protein AMPylation()

door Lewallen, Daniel M., Sreelatha, Anju, Dharmarajan, Venkatasubramanian, Madoux, Franck, Chase, Peter, Griffin, Patrick R., Orth, Kim, Hodder, Peter, Thompson, Paul R.
Gepubliceerd in 2013