A High-Throughput Screening Compatible Assay for Activators and Inhibitors of Methionine Sulfoxide Reductase A

por Brunell, David, Weissbach, Herbert, Hodder, Peter, Brot, Nathan
Publicado 2010

Monitoring of HTS Compound Library Quality via a High-Resolution Image Acquisition and Processing Instrument

por Baillargeon, Pierre, Scampavia, Louis, Einsteder, Ross, Hodder, Peter
Publicado 2011

Synthesis of Small Molecule Inhibitors of the Orphan Nuclear Receptor Steroidogenic Factor-1 (NR5A1) Based on Isoquinolinone Scaffolds

por Roth, Joshua, Madoux, Franck, Hodder, Peter, Roush, William R.
Publicado 2008

Inhibition of Adrenocortical Carcinoma Cell Proliferation by Steroidogenic Factor-1 Inverse Agonists

por Doghman, Mabrouka, Cazareth, Julie, Douguet, Dominique, Madoux, Franck, Hodder, Peter, Lalli, Enzo
Publicado 2009

Dynamics of the formation of a hydrogel by a pathogenic amyloid peptide: islet amyloid polypeptide

por Jean, Létitia, Lee, Chiu Fan, Hodder, Peter, Hawkins, Nick, Vaux, David J.
Publicado en Sci Rep (2016)

Inhibition of Adrenocortical Carcinoma Cell Proliferation by Steroidogenic Factor-1 Inverse Agonists

por Doghman, Mabrouka, Cazareth, Julie, Douguet, Dominique, Madoux, Franck, Hodder, Peter, Lalli, Enzo
Publicado en Mol Endocrinol (2009)

An altered zinc-binding site confers resistance to a covalent inactivator of New Delhi metallo-beta-lactamase-1 (NDM-1) discovered by high-throughput screening

por Thomas, Pei W., Spicer, Timothy, Cammarata, Michael, Brodbelt, Jennifer S., Hodder, Peter, Fast, Walter
Publicado 2013

High Throughput Screen for Pharmacoperones of the Vasopressin Type 2 Receptor

por Conn, P. Michael, Smith, Emery, Hodder, Peter, Janovick, Jo Ann, Smithson, David C.
Publicado 2013

Development of an HTS-Compatible Assay for the Discovery of ASK1 Signalosome Inhibitors Using AlphaScreen Technology

por Sturchler, Emmanuel, Chen, Weimin, Spicer, Timothy, Hodder, Peter, McDonald, Patricia, Duckett, Derek
Publicado 2014

In Pursuit of Synthetic Modulators for the Orphan Retina-Specific Nuclear Receptor NR2E3

por Qin, Qiong, Knapinska, Anna, Dobri, Nicoleta, Madoux, Franck, Chase, Peter, Hodder, Peter, Petrukhin, Konstantin
Publicado 2013

An Ultra-High Throughput Cell-Based Screen for Wee1 Degradation Inhibitors

por MADOUX, FRANCK, SIMANSKI, SCOTT, CHASE, PETER, MISHRA, JITENDRA K., ROUSH, WILLIAM R., AYAD, NAGI G., HODDER, PETER
Publicado 2010

Identification of Novel, Exosite-Binding Matrix Metalloproteinase-13 Inhibitor Scaffolds

por Roth, Joshua, Minond, Dmitriy, Darout, Etzer, Liu, Qin, Lauer, Janelle, Hodder, Peter, Fields, Gregg B., Roush, William R.
Publicado 2011

A FluoPol-ABPP PAD2 High-Throughput Screen Identifies the First Calcium Site Inhibitor Targeting the PADs

por Lewallen, Daniel M., Bicker, Kevin L., Madoux, Franck, Chase, Peter, Anguish, Lynne, Coonrod, Scott, Hodder, Peter, Thompson, Paul R.
Publicado 2014

High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate

por Lauer-Fields, Janelle L., Minond, Dmitriy, Chase, Peter S., Baillargeon, Pierre E., Saldanha, S. Adrian, Stawikowska, Roma, Hodder, Peter, Fields, Gregg B.
Publicado 2008

Screening of potential ADAMTS-4 inhibitors utilizing a collagen-model FRET substrate

por Lauer-Fields, Janelle L., Spicer, Timothy P., Chase, Peter S., Cudic, Mare, Burstein, Gayle D., Nagase, Hideaki, Hodder, Peter, Fields, Gregg B.
Publicado 2007

Discovery, synthesis and SAR analysis of novel selective small molecule S1P(4)–R agonists based on a (2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-one chem...

por Urbano, Mariangela, Guerrero, Miguel, Velaparthi, Subash, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
Publicado 2011

Potent and Selective Inhibitors of Glutathione S-transferase Omega 1 that Impair Cancer Drug Resistance

por Tsuboi, Katsunori, Bachovchin, Daniel A., Speers, Anna E., Spicer, Timothy P., Fernandez-Vega, Virneliz, Hodder, Peter, Rosen, Hugh, Cravatt, Benjamin F.
Publicado 2011

Potent, selective and cell penetrant inhibitors of SF-1 by functional uHTS

por Madoux, Franck, Li, Xiaolin, Chase, Peter, Zastrow, Gina, Cameron, Michael D., Conkright, Juliana J., Griffin, Patrick R., Thacher, Scott, Hodder, Peter
Publicado 2008

Discovery, Design and Synthesis of Novel Potent and Selective Sphingosine-1-Phosphate 4 Receptor (S1P(4)-R) Agonists

por Guerrero, Miguel, Urbano, Mariangela, Zhao, Jian, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
Publicado 2011

Inhibiting AMPylation: A novel screen to identify the first small molecule inhibitors of protein AMPylation()

por Lewallen, Daniel M., Sreelatha, Anju, Dharmarajan, Venkatasubramanian, Madoux, Franck, Chase, Peter, Griffin, Patrick R., Orth, Kim, Hodder, Peter, Thompson, Paul R.
Publicado 2013