A High-Throughput Screening Compatible Assay for Activators and Inhibitors of Methionine Sulfoxide Reductase A

par Brunell, David, Weissbach, Herbert, Hodder, Peter, Brot, Nathan
Publié 2010

Monitoring of HTS Compound Library Quality via a High-Resolution Image Acquisition and Processing Instrument

par Baillargeon, Pierre, Scampavia, Louis, Einsteder, Ross, Hodder, Peter
Publié 2011

Synthesis of Small Molecule Inhibitors of the Orphan Nuclear Receptor Steroidogenic Factor-1 (NR5A1) Based on Isoquinolinone Scaffolds

par Roth, Joshua, Madoux, Franck, Hodder, Peter, Roush, William R.
Publié 2008

Inhibition of Adrenocortical Carcinoma Cell Proliferation by Steroidogenic Factor-1 Inverse Agonists

par Doghman, Mabrouka, Cazareth, Julie, Douguet, Dominique, Madoux, Franck, Hodder, Peter, Lalli, Enzo
Publié 2009

Dynamics of the formation of a hydrogel by a pathogenic amyloid peptide: islet amyloid polypeptide

par Jean, Létitia, Lee, Chiu Fan, Hodder, Peter, Hawkins, Nick, Vaux, David J.
Publié dans Sci Rep (2016)

Inhibition of Adrenocortical Carcinoma Cell Proliferation by Steroidogenic Factor-1 Inverse Agonists

par Doghman, Mabrouka, Cazareth, Julie, Douguet, Dominique, Madoux, Franck, Hodder, Peter, Lalli, Enzo
Publié dans Mol Endocrinol (2009)

An altered zinc-binding site confers resistance to a covalent inactivator of New Delhi metallo-beta-lactamase-1 (NDM-1) discovered by high-throughput screening

par Thomas, Pei W., Spicer, Timothy, Cammarata, Michael, Brodbelt, Jennifer S., Hodder, Peter, Fast, Walter
Publié 2013

High Throughput Screen for Pharmacoperones of the Vasopressin Type 2 Receptor

par Conn, P. Michael, Smith, Emery, Hodder, Peter, Janovick, Jo Ann, Smithson, David C.
Publié 2013

Development of an HTS-Compatible Assay for the Discovery of ASK1 Signalosome Inhibitors Using AlphaScreen Technology

par Sturchler, Emmanuel, Chen, Weimin, Spicer, Timothy, Hodder, Peter, McDonald, Patricia, Duckett, Derek
Publié 2014

In Pursuit of Synthetic Modulators for the Orphan Retina-Specific Nuclear Receptor NR2E3

par Qin, Qiong, Knapinska, Anna, Dobri, Nicoleta, Madoux, Franck, Chase, Peter, Hodder, Peter, Petrukhin, Konstantin
Publié 2013

An Ultra-High Throughput Cell-Based Screen for Wee1 Degradation Inhibitors

par MADOUX, FRANCK, SIMANSKI, SCOTT, CHASE, PETER, MISHRA, JITENDRA K., ROUSH, WILLIAM R., AYAD, NAGI G., HODDER, PETER
Publié 2010

Identification of Novel, Exosite-Binding Matrix Metalloproteinase-13 Inhibitor Scaffolds

par Roth, Joshua, Minond, Dmitriy, Darout, Etzer, Liu, Qin, Lauer, Janelle, Hodder, Peter, Fields, Gregg B., Roush, William R.
Publié 2011

A FluoPol-ABPP PAD2 High-Throughput Screen Identifies the First Calcium Site Inhibitor Targeting the PADs

par Lewallen, Daniel M., Bicker, Kevin L., Madoux, Franck, Chase, Peter, Anguish, Lynne, Coonrod, Scott, Hodder, Peter, Thompson, Paul R.
Publié 2014

High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate

par Lauer-Fields, Janelle L., Minond, Dmitriy, Chase, Peter S., Baillargeon, Pierre E., Saldanha, S. Adrian, Stawikowska, Roma, Hodder, Peter, Fields, Gregg B.
Publié 2008

Screening of potential ADAMTS-4 inhibitors utilizing a collagen-model FRET substrate

par Lauer-Fields, Janelle L., Spicer, Timothy P., Chase, Peter S., Cudic, Mare, Burstein, Gayle D., Nagase, Hideaki, Hodder, Peter, Fields, Gregg B.
Publié 2007

Discovery, synthesis and SAR analysis of novel selective small molecule S1P(4)–R agonists based on a (2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-one chem...

par Urbano, Mariangela, Guerrero, Miguel, Velaparthi, Subash, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
Publié 2011

Potent and Selective Inhibitors of Glutathione S-transferase Omega 1 that Impair Cancer Drug Resistance

par Tsuboi, Katsunori, Bachovchin, Daniel A., Speers, Anna E., Spicer, Timothy P., Fernandez-Vega, Virneliz, Hodder, Peter, Rosen, Hugh, Cravatt, Benjamin F.
Publié 2011

Potent, selective and cell penetrant inhibitors of SF-1 by functional uHTS

par Madoux, Franck, Li, Xiaolin, Chase, Peter, Zastrow, Gina, Cameron, Michael D., Conkright, Juliana J., Griffin, Patrick R., Thacher, Scott, Hodder, Peter
Publié 2008

Discovery, Design and Synthesis of Novel Potent and Selective Sphingosine-1-Phosphate 4 Receptor (S1P(4)-R) Agonists

par Guerrero, Miguel, Urbano, Mariangela, Zhao, Jian, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
Publié 2011

Inhibiting AMPylation: A novel screen to identify the first small molecule inhibitors of protein AMPylation()

par Lewallen, Daniel M., Sreelatha, Anju, Dharmarajan, Venkatasubramanian, Madoux, Franck, Chase, Peter, Griffin, Patrick R., Orth, Kim, Hodder, Peter, Thompson, Paul R.
Publié 2013