Modulators of the Sphingosine 1-Phosphate Receptor 1

מאת Urbano, Mariangela, Guerrero, Miguel, Rosen, Hugh, Roberts, Edward
יצא לאור 2013

SAR analysis of novel non-peptidic NPBWR1 (GPR7) antagonists

מאת Guerrero, Miguel, Urbano, Mariangela, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
יצא לאור 2012

Discovery, Design and Synthesis of the First Reported Potent and Selective Sphingosine-1-Phosphate 4 (S1P(4)) Receptor Antagonists

מאת Guerrero, Miguel, Urbano, Mariangela, Velaparthi, Subash, Zhao, Jian, Schaeffer, MarieTherese, Brown, Steve, Rosen, Hugh, Roberts, Edward
יצא לאור 2011

SAR Analysis of Innovative Selective Small Molecule Antagonists of Sphingosine-1-Phosphate 4 (S1P(4)) Receptor

מאת Urbano, Mariangela, Guerrero, Miguel, Zhao, Jian, Velaparthi, Subash, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
יצא לאור 2011

Discovery, synthesis and SAR analysis of novel selective small molecule S1P(4)–R agonists based on a (2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-one chem...

מאת Urbano, Mariangela, Guerrero, Miguel, Velaparthi, Subash, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
יצא לאור 2011

Discovery, Design and Synthesis of Novel Potent and Selective Sphingosine-1-Phosphate 4 Receptor (S1P(4)-R) Agonists

מאת Guerrero, Miguel, Urbano, Mariangela, Zhao, Jian, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
יצא לאור 2011

Discovery, design and synthesis of a selective S1P(3) receptor allosteric agonist

מאת Guerrero, Miguel, Poddutoori, Ramulu, Urbano, Mariangela, Peng, Xuemei, Spicer, Timothy P., Chase, Peter S., Hodder, Peter S., Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
יצא לאור 2013

Design, synthesis and SAR analysis of novel potent and selective small molecule antagonists of NPBWR1 (GPR7)

מאת Urbano, Mariangela, Guerrero, Miguel, Zhao, Jian, Velaparthi, Subash, Saldanha, S. Adrian, Chase, Peter, Wang, Zhiwei, Civelli, Olivier, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward
יצא לאור 2012

Design and Synthesis of a Novel and Selective Kappa Opioid Receptor (KOR) Antagonist (BTRX-335140)

מאת Guerrero, Miguel, Urbano, Mariangela, Kim, Eun-Kyong, Gamo, Ana M., Riley, Sean, Abgaryan, Lusine, Leaf, Nora, Van Orden, Lori Jean, Brown, Steven J., Xie, Jennifer Y., Porreca, Frank, Cameron, Michael D., Rosen, Hugh, Roberts, Edward
הוצא לאור ב J Med Chem (2019)