Resultados da pesquisa por Autor

1

HIV-1 IN Inhibitors: 2010 Update and Perspectives

HIV-1 IN Inhibitors: 2010 Update and Perspectives

Por Marchand, Christophe, Maddali, Kasthuraiah, Metifiot, Mathieu, Pommier, Yves
Publicado em 2009

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2

Resistance to Integrase Inhibitors

Resistance to Integrase Inhibitors

Por Métifiot, Mathieu, Marchand, Christophe, Maddali, Kasthuraiah, Pommier, Yves
Publicado em 2010

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3

Role of tyrosyl-DNA phosphodiesterase (TDP1) in mitochondria

Role of tyrosyl-DNA phosphodiesterase (TDP1) in mitochondria

Por Das, Benu Brata, Dexheimer, Thomas S., Maddali, Kasthuraiah, Pommier, Yves
Publicado em 2010

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4

Diketoacid – Genre HIV-1 Integrase Inhibitors Containing Enantiomeric Arylamide Functionality

Diketoacid – Genre HIV-1 Integrase Inhibitors Containing Enantiomeric Arylamide Functionality

Por Zhao, Xue Zhi, Maddali, Kasthuraiah, Marchand, Christophe, Pommier, Yves, Burke, Terrence R.
Publicado em 2009

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5

Biochemical and Pharmacological Analyses of HIV-1 Integrase Flexible Loop Mutants Resistant To Raltegravir

Biochemical and Pharmacological Analyses of HIV-1 Integrase Flexible Loop Mutants Resistant To Raltegravir

Por Métifiot, Mathieu, Maddali, Kasthuraiah, Naumova, Alena, Zhang, Xuemin, Marchand, Christophe, Pommier, Yves
Publicado em 2010

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6

3-Hydroxypyrimidine-2,4-diones as an Inhibitor Scaffold of HIV Integrase

3-Hydroxypyrimidine-2,4-diones as an Inhibitor Scaffold of HIV Integrase

Por Tang, Jing, Maddali, Kasthuraiah, Sham, Yuk Y., Vince, Robert, Pommier, Yves, Wang, Zhengqiang
Publicado em 2011

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7

6-Benzoyl-3-hydroxypyrimidine-2,4-diones as Dual Inhibitors of HIV Reverse Transcriptase and Integrase

6-Benzoyl-3-hydroxypyrimidine-2,4-diones as Dual Inhibitors of HIV Reverse Transcriptase and Integrase

Por Tang, Jing, Maddali, Kasthuraiah, Dreis, Christine D., Sham, Yuk Y., Vince, Robert, Pommier, Yves, Wang, Zhengqiang
Publicado em 2011

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8

N-3 Hydroxylation of Pyrimidine-2,4-diones Yields Dual Inhibitors of HIV Reverse Transcriptase and Integrase

N-3 Hydroxylation of Pyrimidine-2,4-diones Yields Dual Inhibitors of HIV Reverse Transcriptase and Integrase

Por Tang, Jing, Maddali, Kasthuraiah, Dreis, Christine D., Sham, Yuk Y., Vince, Robert, Pommier, Yves, Wang, Zhengqiang
Publicado em 2010

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9

Examination of halogen substituent effects on HIV-1 integrase inhibitors derived from 2,3-dihydro-6,7-dihydroxy-1H-isoindol-1-ones and 4,5-dihydroxy-1H-isoindole-1,3(2H)-diones

Examination of halogen substituent effects on HIV-1 integrase inhibitors derived from 2,3-dihydro-6,7-dihydroxy-1H-isoindol-1-ones and 4,5-dihydroxy-1H-isoindole-1,3(2H)-diones

Por Zhao, Xue Zhi, Maddali, Kasthuraiah, Vu, B. Christie, Marchand, Christophe, Hughes, Stephen H., Pommier, Yves, Burke, Terrence R.
Publicado em 2009

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10

Probing chelation motifs in HIV integrase inhibitors

Probing chelation motifs in HIV integrase inhibitors

Por Agrawal, Arpita, DeSoto, Jamie, Fullagar, Jessica L., Maddali, Kasthuraiah, Rostami, Shahrzad, Richman, Douglas D., Pommier, Yves, Cohen, Seth M.
Publicado em 2012

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11

Development of Tricyclic Hydroxy-1H-pyrrolopyridine-trione Containing HIV-1 Integrase Inhibitors

Development of Tricyclic Hydroxy-1H-pyrrolopyridine-trione Containing HIV-1 Integrase Inhibitors

Por Zhao, Xue Zhi, Maddali, Kasthuraiah, Metifiot, Mathieu, Smith, Steven J., Vu, B. Christie, Marchand, Christophe, Hughes, Stephen H., Pommier, Yves, Burke, Terrence R.
Publicado em 2011

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12

6,7-Dihydroxy-1-oxoisoindoline-4-sulfonamide-containing HIV-1 Integrase Inhibitors

6,7-Dihydroxy-1-oxoisoindoline-4-sulfonamide-containing HIV-1 Integrase Inhibitors

Por Zhao, Xue Zhi, Maddali, Kasthuraiah, Smith, Steven J., Métifiot, Mathieu, Johnson, Barry C., Marchand, Christophe, Hughes, Stephen H., Pommier, Yves, Burke, Terrence R.
Publicado em 2012

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13

Activities, crystal structures and molecular dynamics of dihydro-1H-isoindole derivatives, inhibitors of HIV-1 integrase

Activities, crystal structures and molecular dynamics of dihydro-1H-isoindole derivatives, inhibitors of HIV-1 integrase

Por Métifiot, Mathieu, Maddali, Kasthuraiah, Johnson, Barry C., Hare, Stephen, Smith, Steven J., Zhao, XueZhi, Marchand, Christophe, Burke, Terrence R., Hughes, Stephen H., Cherepanov, Peter, Pommier, Yves
Publicado em 2012

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14

Peptidic HIV integrase inhibitors derived from HIV gene products: structure-activity relationship studies

Peptidic HIV integrase inhibitors derived from HIV gene products: structure-activity relationship studies

Por Suzuki, Shintaro, Maddali, Kasthuraiah, Hashimoto, Chie, Urano, Emiko, Ohashi, Nami, Tanaka, Tomohiro, Ozaki, Taro, Arai, Hiroshi, Tsutsumi, Hiroshi, Narumi, Tetsuo, Nomura, Wataru, Yamamoto, Naoki, Pommier, Yves, Komano, Jun A., Tamamura, Hirokazu
Publicado no Bioorg Med Chem (2010)

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15

Peptide HIV-1 Integrase Inhibitors from HIV-1 Gene Products

Peptide HIV-1 Integrase Inhibitors from HIV-1 Gene Products

Por Suzuki, Shintaro, Urano, Emiko, Hashimoto, Chie, Tsutsumi, Hiroshi, Nakahara, Toru, Tanaka, Tomohiro, Nakanishi, Yuta, Maddali, Kasthuraiah, Han, Yan, Hamatake, Makiko, Miyauchi, Kosuke, Pommier, Yves, Beutler, John A., Sugiura, Wataru, Fuji, Hideyoshi, Hoshino, Tyuji, Itotani, Kyoko, Nomura, Wataru, Narumi, Tetsuo, Yamamoto, Naoki, Komano, Jun A., Tamamura, Hirokazu
Publicado no J Med Chem (2010)

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16

Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase

Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase

Por Costi, Roberta, Métifiot, Mathieu, Chung, Suhman, Cuzzucoli Crucitti, Giuliana, Maddali, Kasthuraiah, Pescatori, Luca, Messore, Antonella, Madia, Valentina Noemi, Pupo, Giovanni, Scipione, Luigi, Tortorella, Silvano, Di Leva, Francesco Saverio, Cosconati, Sandro, Marinelli, Luciana, Novellino, Ettore, Le Grice, Stuart F. J., Corona, Angela, Pommier, Yves, Marchand, Christophe, Di Santo, Roberto
Publicado em 2014

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