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Probing chelation motifs in HIV integrase inhibitors

A series of HIV integrase (HIV-1 IN) inhibitors were synthesized to evaluate the role of the metal-binding group (MBG) in this class of metalloenzyme inhibitors. A total of 21 different raltegravir-chelator derivative (RCD) compounds were prepared that differed only in the nature of the MBG. These I...

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Bibliografiske detaljer
Main Authors: Agrawal, Arpita, DeSoto, Jamie, Fullagar, Jessica L., Maddali, Kasthuraiah, Rostami, Shahrzad, Richman, Douglas D., Pommier, Yves, Cohen, Seth M.
Format: Artigo
Sprog:Inglês
Udgivet: National Academy of Sciences 2012
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Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3289312/
https://ncbi.nlm.nih.gov/pubmed/22308350
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1112389109
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