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3-Hydroxypyrimidine-2,4-diones as an Inhibitor Scaffold of HIV Integrase
Integrase (IN) represents a clinically validated target for the development of antivirals against human immunodeficiency virus (HIV). Inhibitors with a novel structure core are essential for combating resistance associated with known IN inhibitors (INIs). We have previously disclosed a novel dual in...
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| Autori principali: | , , , , , |
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| Natura: | Artigo |
| Lingua: | Inglês |
| Pubblicazione: |
2011
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| Soggetti: | |
| Accesso online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3072462/ https://ncbi.nlm.nih.gov/pubmed/21381765 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm1014378 |
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