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Resistance to Integrase Inhibitors

Integrase (IN) is a clinically validated target for the treatment of human immunodeficiency virus infections and raltegravir exhibits remarkable clinical activity. The next most advanced IN inhibitor is elvitegravir. However, mutant viruses lead to treatment failure and mutations within the IN codin...

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Detalhes bibliográficos
Main Authors: Métifiot, Mathieu, Marchand, Christophe, Maddali, Kasthuraiah, Pommier, Yves
Formato: Artigo
Idioma:Inglês
Publicado em: Molecular Diversity Preservation International (MDPI) 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2920056/
https://ncbi.nlm.nih.gov/pubmed/20706558
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/v2071347
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