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Elvitegravir overcomes resistance to raltegravir induced by integrase mutation Y143
OBJECTIVE: In this study, we characterized elvitegravir activity in the context of raltegravir resistance mutations. DESIGN: Using site-directed mutagenesis, we generated recombinant integrase proteins and viruses harboring raltegravir resistance mutation to assess the biochemical and cellular activ...
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| Publicat a: | AIDS |
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| Autors principals: | , , , , , , , |
| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
2011
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7380719/ https://ncbi.nlm.nih.gov/pubmed/21505303 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1097/QAD.0b013e3283473599 |
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