Playing Well with Others! Initiating and sustaining successful collaborations between Industry, Academia and Government

Por Thomas, Craig J., McKew, John C.
Publicado no Curr Top Med Chem (2014)

Synthesis of Substituted 2-phenylhistamines via a Microwave Promoted Suzuki Coupling

Por Skoumbourdis, Amanda P., Moore, Susanna, Landsman, Marc, Thomas, Craig J.
Publicado em 2007

Synthesis of Oxadiazole-2-oxide Analogues as Potential Antischistosomal Agents

Por Rai, Ganesha, Thomas, Craig J., Leister, William, Maloney, David J.
Publicado em 2009

Chiral Kinase Inhibitors

Por Jiang, Jian-kang, Shen, Min, Thomas, Craig J., Boxer, Mathew B.
Publicado em 2011

Design and synthesis of new bicyclic diketopiperazines as scaffolds for receptor probes of structurally diverse functionality()

Por Besada, Pedro, Mamedova, Liaman, Thomas, Craig J., Costanzi, Stefano, Jacobson, Kenneth A.
Publicado em 2005

Selecting, Acquiring, and Using Small Molecule Libraries for High-Throughput Screening

Por Dandapani, Sivaraman, Rosse, Gerard, Southall, Noel, Salvino, Joseph M., Thomas, Craig J.
Publicado no Curr Protoc Chem Biol (2012)

PfCRT and PfMDR1 modulate interactions of artemisinin derivatives and ion channel blockers

Por Eastman, Richard T., Khine, Pwint, Huang, Ruili, Thomas, Craig J., Su, Xin-zhuan
Publicado no Sci Rep (2016)

Comparison of Raltegravir and Elvitagravir on HIV-1 Integrase Catalytic Reactions and on a Series of Drug-Resistant Integrase Mutants

Por Marinello, Jessica, Marchand, Christophe, Mott, Bryan, Bain, Anjali, Thomas, Craig J., Pommier, Yves
Publicado em 2008

Total synthesis of LL-Z1640-2 utilizing a late-stage intramolecular Nozaki-Hiyama-Kishi reaction

Por LeClair, Christopher A., Boxer, Matthew B., Thomas, Craig J., Maloney, David J.
Publicado em 2010

A Small Molecule Inverse Agonist for the Human Thyroid-Stimulating Hormone Receptor

Por Neumann, Susanne, Huang, Wenwei, Eliseeva, Elena, Titus, Steve, Thomas, Craig J., Gershengorn, Marvin C.
Publicado em 2010

Identification of Oxadiazoles as New Drug Leads for the Control of Schistosomiasis

Por Sayed, Ahmed A., Simeonov, Anton, Thomas, Craig J., Inglese, James, Austin, Christopher P., Williams, David L.
Publicado em 2008

Comparison of Bioluminescent Kinase Assays Using Substrate Depletion and Product Formation

Por Tanega, Cordelle, Shen, Min, Mott, Bryan T., Thomas, Craig J., MacArthur, Ryan, Inglese, James, Auld, Douglas S.
Publicado em 2009

Comprehensive Survey of Chemical Libraries for Drug Discovery and Chemical Biology: 2009

Por Dolle, Roland E., Le Bourdonnec, Bertrand, Worm, Karin, Morales, Guillermo A., Thomas, Craig J., Zhang, Wei
Publicado em 2010

N(4)-Phenyl Modifications of N(2)-(2-hydroxyl)ethyl-6-(pyrrolidin-1-yl)-1,3,5-triazine-2,4-diamines Enhance Glucocerebrosidase Inhibition by Small Molecules with Potential as Chemi...

Por Huang, Wenwei, Zheng, Wei, Urban, Daniel J., Inglese, James, Sidransky, Ellen, Austin, Christopher P., Thomas, Craig J.
Publicado em 2007

Proteasome Inactivation Promotes p38 Mitogen-activated Protein Kinase-dependent Phosphatidylinositol 3-kinase Activation and Increases Interleukin-8 Production in Retinal Pigment E...

Por Fernandes, Alexandre F., Bian, Qingning, Jiang, Jian-Kang, Thomas, Craig J., Taylor, Allen, Pereira, Paulo, Shang, Fu
Publicado em 2009

Drug resistant integrase mutants cause aberrant HIV integrations

Por Varadarajan, Janani, McWilliams, Mary Jane, Mott, Bryan T., Thomas, Craig J., Smith, Steven J., Hughes, Stephen H.
Publicado no Retrovirology (2016)

Identification of potent Yes1 kinase inhibitors using a library screening approach

Por Patel, Paresma R., Sun, Hongmao, Li, Samuel Q., Shen, Min, Khan, Javed, Thomas, Craig J., Davis, Mindy I.
Publicado em 2013

Synthesis and N-Methyl-D-aspartate (NMDA) Receptor Activity of Ketamine Metabolites

Por Morris, Patrick J., Moaddel, Ruin, Zanos, Panos, Moore, Curtis E., Gould, Todd, Zarate, Carlos A., Thomas, Craig J.
Publicado no Org Lett (2017)

A Highly Potent and Selective Caspase 1 Inhibitor that Utilizes a Key 3-Cyanopropanoic Acid Moiety

Por Boxer, Matthew B., Quinn, Amy M., Shen, Min, Jadhav, Ajit, Leister, William, Simeonov, Anton, Auld, Douglas S., Thomas, Craig J.
Publicado em 2010

A bi-directional, iterative approach to the structural delineation of the functional “chemoprint” in GPR40 for agonist recognition

Por Tikhonova, Irina G., Sum, Chi Shing, Neumann, Susanne, Thomas, Craig J., Raaka, Bruce M., Costanzi, Stefano, Gershengorn, Marvin C.
Publicado em 2007