Human TSH receptor ligands as pharmacological probes with potential clinical application

af Neumann, Susanne, Raaka, Bruce M, Gershengorn, Marvin C
Udgivet 2009

Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor

af Thirunarayanan, Nanthakumar, Raaka, Bruce M., Gershengorn, Marvin C.
Udgivet 2012

Constitutively Active Thyrotropin And Thyrotropin-Releasing Hormone Receptors And Their Inverse Agonists

af Neumann, Susanne, Raaka, Bruce M., Gershengorn, Marvin C.
Udgivet i Methods Enzymol (2010)

Rational discovery of novel nuclear hormone receptor antagonists

af Schapira, Matthieu, Raaka, Bruce M., Samuels, Herbert H., Abagyan, Ruben
Udgivet 2000

In silico discovery of novel Retinoic Acid Receptor agonist structures

af Schapira, Matthieu, Raaka, Bruce M, Samuels, Herbert H, Abagyan, Ruben
Udgivet 2001

Thyrotropin-Releasing Hormone Receptor Type 1 (TRH-R1), not TRH-R2, Primarily Mediates Taltirelin Actions in the CNS of Mice

af Thirunarayanan, Nanthakumar, Nir, Eshel A, Raaka, Bruce M, Gershengorn, Marvin C
Udgivet 2013

High Levels of TRH Receptors Activate Programmed Cell Death in Human Pancreatic Precursors

af Mulla, Christopher M., Geras-Raaka, Elizabeth, Raaka, Bruce M., Gershengorn, Marvin C.
Udgivet 2009

TRH Receptor Type 2 Deficient Mice are Euthyroid and Exhibit Increased Depression and Reduced Anxiety Phenotypes

af Sun, Yuhua, Zupan, Bojana, Raaka, Bruce M., Toth, Miklos, Gershengorn, Marvin C.
Udgivet 2008

Erythropoietin Signaling: A Novel Regulator of White Adipose Tissue Inflammation During Diet-Induced Obesity

af Alnaeeli, Mawadda, Raaka, Bruce M., Gavrilova, Oksana, Teng, Ruifeng, Chanturiya, Tatyana, Noguchi, Constance Tom
Udgivet 2014

Human pancreatic precursor cells secrete FGF2 to stimulate clustering into hormone-expressing islet-like cell aggregates

af Hardikar, Anandwardhan A., Marcus-Samuels, Bernice, Geras-Raaka, Elizabeth, Raaka, Bruce M., Gershengorn, Marvin C.
Udgivet 2003

Endocrine Precursor Cells from Mouse Islets Are Not Generated by Epithelial-to-Mesenchymal Transition of Mature Beta Cells

af Morton, Russell A., Geras-Raaka, Elizabeth, Wilson, Leah M., Raaka, Bruce M., Gershengorn, Marvin C.
Udgivet 2007

Evidence for cooperative signal triggering at the extracellular loops of the TSH receptor

af Kleinau, Gunnar, Jaeschke, Holger, Mueller, Sandra, Raaka, Bruce M., Neumann, Susanne, Paschke, Ralf, Krause, Gerd
Udgivet 2008

A Drug-Like Antagonist Inhibits Thyrotropin Receptor–Mediated Stimulation of cAMP Production in Graves' Orbital Fibroblasts

af Neumann, Susanne, Pope, Arthur, Geras-Raaka, Elizabeth, Raaka, Bruce M., Bahn, Rebecca S., Gershengorn, Marvin C.
Udgivet 2012

Perilipin family members preferentially sequester to either triacylglycerol-specific or cholesteryl-ester-specific intracellular lipid storage droplets

af Hsieh, Kai, Lee, Yun Kyung, Londos, Constantine, Raaka, Bruce M., Dalen, Knut Tomas, Kimmel, Alan R.
Udgivet 2012

Insulin but Not Glucagon Gene is Silenced in Human Pancreas-Derived Mesenchymal Stem Cells

af Wilson, Leah M., Wong, Stephen H.K., Yu, Ningpu, Geras-Raaka, Elizabeth, Raaka, Bruce M., Gershengorn, Marvin C.
Udgivet 2009

Discovery of novel agonists and antagonists of the free fatty acid receptor one (FFAR1) using virtual screening

af Tikhonova, Irina G., Sum, Chi Shing, Neumann, Susanne, Engel, Stanislav, Raaka, Bruce M., Costanzi, Stefano, Gershengorn, Marvin C.
Udgivet 2008

A bi-directional, iterative approach to the structural delineation of the functional “chemoprint” in GPR40 for agonist recognition

af Tikhonova, Irina G., Sum, Chi Shing, Neumann, Susanne, Thomas, Craig J., Raaka, Bruce M., Costanzi, Stefano, Gershengorn, Marvin C.
Udgivet 2007

Discovery of diverse thyroid hormone receptor antagonists by high-throughput docking

af Schapira, Matthieu, Raaka, Bruce M., Das, Sharmistha, Fan, Li, Totrov, Maxim, Zhou, Zhiguo, Wilson, Stephen R., Abagyan, Ruben, Samuels, Herbert H.
Udgivet 2003

A Low-Molecular-Weight Antagonist for the Human Thyrotropin Receptor with Therapeutic Potential for Hyperthyroidism

af Neumann, Susanne, Kleinau, Gunnar, Costanzi, Stefano, Moore, Susanna, Jiang, Jian-kang, Raaka, Bruce M., Thomas, Craig J., Krause, Gerd, Gershengorn, Marvin C.
Udgivet 2008

Evaluation of gene expression measurements from commercial microarray platforms

af Tan, Paul K., Downey, Thomas J., Spitznagel, Edward L., Xu, Pin, Fu, Dadin, Dimitrov, Dimiter S., Lempicki, Richard A., Raaka, Bruce M., Cam, Margaret C.
Udgivet 2003