Development of homogeneous luminescence assays for histone demethylase catalysis and binding

ανά Kawamura, Akane, Tumber, Anthony, Rose, Nathan R., King, Oliver N. F., Daniel, Michelle, Oppermann, Udo, Heightman, Tom D., Schofield, Christopher
Τόπος έκδοσης Anal Biochem (2010)

Large-Scale Structural Analysis of the Classical Human Protein Tyrosine Phosphatome

ανά Barr, Alastair J., Ugochukwu, Emilie, Lee, Wen Hwa, King, Oliver N.F., Filippakopoulos, Panagis, Alfano, Ivan, Savitsky, Pavel, Burgess-Brown, Nicola A., Müller, Susanne, Knapp, Stefan
Έκδοση 2009

Inhibition of Histone Demethylases by 4-Carboxy-2,2′-Bipyridyl Compounds

ανά Chang, Kai-Hsuan, King, Oliver N.F., Tumber, Anthony, Woon, Esther C.Y., Heightman, Tom D., McDonough, Michael A., Schofield, Christopher J., Rose, Nathan R.
Τόπος έκδοσης ChemMedChem (2011)

Selective Inhibitors of the JMJD2 Histone Demethylases: Combined Nondenaturing Mass Spectrometric Screening and Crystallographic Approaches

ανά Rose, Nathan R., Woon, Esther C. Y., Kingham, Guy L., King, Oliver N. F., Mecinović, Jasmin, Clifton, Ian J., Ng, Stanley S., Talib-Hardy, Jobina, Oppermann, Udo, McDonough, Michael A., Schofield, Christopher J.
Έκδοση 2010

Quantitative High-Throughput Screening Identifies 8-Hydroxyquinolines as Cell-Active Histone Demethylase Inhibitors

ανά King, Oliver N. F., Li, Xuan Shirley, Sakurai, Masaaki, Kawamura, Akane, Rose, Nathan R., Ng, Stanley S., Quinn, Amy M., Rai, Ganesha, Mott, Bryan T., Beswick, Paul, Klose, Robert J., Oppermann, Udo, Jadhav, Ajit, Heightman, Tom D., Maloney, David J., Schofield, Christopher J., Simeonov, Anton
Έκδοση 2010

Highly selective inhibition of histone demethylases by de novo macrocyclic peptides

ανά Kawamura, Akane, Münzel, Martin, Kojima, Tatsuya, Yapp, Clarence, Bhushan, Bhaskar, Goto, Yuki, Tumber, Anthony, Katoh, Takayuki, King, Oliver N. F., Passioura, Toby, Walport, Louise J., Hatch, Stephanie B., Madden, Sarah, Müller, Susanne, Brennan, Paul E., Chowdhury, Rasheduzzaman, Hopkinson, Richard J., Suga, Hiroaki, Schofield, Christopher J.
Τόπος έκδοσης Nat Commun (2017)

The Plant Growth Regulator Daminozide is a Selective Inhibitor of the Human KDM2/7 Histone Demethylases

ανά Rose, Nathan R., Woon, Esther C.Y., Tumber, Anthony, Walport, Louise J., Chowdhury, Rasheduzzaman, Li, Xuan Shirley, King, Oliver N.F., Lejeune, Clarisse, Ng, Stanley S., Krojer, Tobias, Chan, Mun Chiang, Rydzik, Anna M., Hopkinson, Richard J., Che, Ka Hing, Daniel, Michelle, Strain-Damerell, Claire, Gileadi, Carina, Kochan, Grazyna, Leung, Ivanhoe K. H., Dunford, James, Yeoh, Kar Kheng, Ratcliffe, Peter J., Burgess-Brown, Nicola, von Delft, Frank, Muller, Susanne, Marsden, Brian, Brennan, Paul E., McDonough, Michael A., Oppermann, Udo, Klose, Robert J., Schofield, Christopher J., Kawamura, Akane
Τόπος έκδοσης J Med Chem (2012)

5-Carboxy-8-hydroxyquinoline is a Broad Spectrum 2-Oxoglutarate Oxygenase Inhibitor which Causes Iron Translocation

ανά Hopkinson, Richard J., Tumber, Anthony, Yapp, Clarence, Chowdhury, Rasheduzzaman, Aik, WeiShen, Che, Ka Hing, Li, Xuan Shirley, Kristensen, Jan B. L., King, Oliver N. F., Chan, Mun Chiang, Yeoh, Kar Kheng, Choi, Hwanho, Walport, Louise J., Thinnes, Cyrille C., Bush, Jacob T., Lejeune, Clarisse, Rydzik, Anna M., Rose, Nathan R., Bagg, Eleanor A., McDonough, Michael A., Krojer, Tobias, Yue, Wyatt W., Ng, Stanley S., Olsen, Lars, Brennan, Paul E., Oppermann, Udo, Muller-Knapp, Susanne, Klose, Robert J., Ratcliffe, Peter J., Schofield, Christopher J., Kawamura, Akane
Τόπος έκδοσης Chem Sci (2013)