ABCG2 is not able to catalyze glutathione efflux and does not contribute to GSH-dependent collateral sensitivity

Por Gauthier, Charlotte, Ozvegy-Laczka, Csilla, Szakacs, Gergely, Sarkadi, Balazs, Di Pietro, Attilio
Publicado em 2013

Localization of putative binding sites for cyclic guanosine monophosphate and the anti-cancer drug 5-fluoro-2′-deoxyuridine-5′-monophosphate on ABCC11 in silico models

Por Honorat, Mylène, Terreux, Raphaël, Falson, Pierre, Di Pietro, Attilio, Dumontet, Charles, Payen, Lea
Publicado em 2013

ABCG2 Transports and Transfers Heme to Albumin through Its Large Extracellular Loop

Por Desuzinges-Mandon, Elodie, Arnaud, Ophélie, Martinez, Lorena, Huché, Frédéric, Di Pietro, Attilio, Falson, Pierre
Publicado em 2010

Microparticle-Mediated Transfer of the Viral Receptors CAR and CD46, and the CFTR Channel in a CHO Cell Model Confers New Functions to Target Cells

Por Gonzalez, Gaëlle, Vituret, Cyrielle, Di Pietro, Attilio, Chanson, Marc, Boulanger, Pierre, Hong, Saw-See
Publicado em 2012

Flavonoids: A class of modulators with bifunctional interactions at vicinal ATP- and steroid-binding sites on mouse P-glycoprotein

Por Conseil, Gwenaelle, Baubichon-Cortay, Helene, Dayan, Guila, Jault, Jean-Michel, Barron, Denis, Di Pietro, Attilio
Publicado em 1998

MRP8/ABCC11 Expression Is Regulated by Dexamethasone in Breast Cancer Cells and Is Associated to Progesterone Receptor Status in Breast Tumors

Por Honorat, Mylène, Mesnier, Aurélia, Vendrell, Julie, Di Pietro, Attilio, Lin, Valérie, Dumontet, Charles, Cohen, Pascale, Payen, Léa
Publicado em 2011

Targeting the Achilles Heel of Multidrug-Resistant Cancer by Exploiting the Fitness Cost of Resistance

Por Szakács, Gergely, Hall, Matthew D., Gottesman, Michael M., Boumendjel, Ahcène, Kachadourian, Remy, Day, Brian J., Baubichon-Cortay, Hélène, Di Pietro, Attilio
Publicado em 2014

A Synthetic Chalcone as a Potent Inducer of Glutathione Biosynthesis

Por Kachadourian, Remy, Day, Brian J., Pugazhenti, Subbiah, Franklin, Christopher C., Genoux-Bastide, Estelle, Mahaffey, Gregory, Gauthier, Charlotte, Di Pietro, Attilio, Boumendjel, Ahcène
Publicado em 2012

High-Affinity Binding of Silybin Derivatives to the Nucleotide-Binding Domain of a Leishmania tropica P-Glycoprotein-Like Transporter and Chemosensitization of a Multidrug-Resistan...

Por Pérez-Victoria, José M., Pérez-Victoria, F. Javier, Conseil, Gwenaëlle, Maitrejean, Mathias, Comte, Gilles, Barron, Denis, Di Pietro, Attilio, Castanys, Santiago, Gamarro, Francisco
Publicado em 2001

The ABC transporter BmrA from Bacillus subtilis is a functional dimer when in a detergent-solubilized state

Por Ravaud, Stéphanie, Do Cao, Marie-Ange, Jidenko, Marie, Ebel, Christine, Le Maire, Marc, Jault, Jean-Michel, Di Pietro, Attilio, Haser, Richard, Aghajari, Nushin
Publicado em 2006

Becatecarin (rebeccamycin analog, NSC 655649) is a transport substrate and induces expression of the ATP-binding cassette transporter, ABCG2, in lung carcinoma cells

Por Robey, Robert W., Obrzut, Tomasz, Shukla, Suneet, Polgar, Orsolya, Macalou, Sira, Bahr, Julian C., Di Pietro, Attilio, Ambudkar, Suresh V., Bates, Susan E.
Publicado em 2009

Investigation of Chalcones as Selective Inhibitors of the Breast Cancer Resistance Protein: Critical Role of Methoxylation in both Inhibition Potency and Cytotoxicity

Por Valdameri, Glaucio, Gauthier, Charlotte, Terreux, Raphaël, Kachadourian, Rémy, Day, Brian J., Winnischofer, Sheila M. B., Rocha, Maria E. M., Frachet, Véronique, Ronot, Xavier, Di Pietro, Attilio, Boumendjel, Ahcène
Publicado em 2012

MBL-II-141, a chromone derivative, enhances irinotecan (CPT-11) anticancer efficiency in ABCG2-positive xenografts

Por Honorat, Mylène, Guitton, Jérôme, Gauthier, Charlotte, Bouard, Charlotte, Lecerf-Schmidt, Florine, Peres, Basile, Terreux, Raphaël, Gervot, Héloïse, Rioufol, Catherine, Boumendjel, Ahcène, Puisieux, Alain, Di Pietro, Attilio, Payen, Léa
Publicado no Oncotarget (2015)

Structuring Detergents for Extracting and Stabilizing Functional Membrane Proteins

Por Matar-Merheb, Rima, Rhimi, Moez, Leydier, Antoine, Huché, Frédéric, Galián, Carmen, Desuzinges-Mandon, Elodie, Ficheux, Damien, Flot, David, Aghajari, Nushin, Kahn, Richard, Di Pietro, Attilio, Jault, Jean-Michel, Coleman, Anthony W., Falson, Pierre
Publicado em 2011

Combination of Suboptimal Doses of Inhibitors Targeting Different Domains of LtrMDR1 Efficiently Overcomes Resistance of Leishmania spp. to Miltefosine by Inhibiting Drug Efflux

Por Pérez-Victoria, José M., Cortés-Selva, Fernando, Parodi-Talice, Adriana, Bavchvarov, Boris I., Pérez-Victoria, F. Javier, Muñoz-Martínez, Francisco, Maitrejean, Mathias, Costi, M. Paola, Barron, Denis, Di Pietro, Attilio, Castanys, Santiago, Gamarro, Francisco
Publicado em 2006

Quinoxaline-substituted chalcones as new inhibitors of breast cancer resistance protein ABCG2: polyspecificity at B-ring position

Por Winter, Evelyn, Gozzi, Gustavo Jabor, Chiaradia-Delatorre, Louise Domeneghini, Daflon-Yunes, Nathalia, Terreux, Raphael, Gauthier, Charlotte, Mascarello, Alessandra, Leal, Paulo César, Cadena, Silvia M, Yunes, Rosendo Augusto, Nunes, Ricardo José, Creczynski-Pasa, Tania Beatriz, Di Pietro, Attilio
Publicado em 2014

Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity

Por Gozzi, Gustavo Jabor, Bouaziz, Zouhair, Winter, Evelyn, Daflon-Yunes, Nathalia, Honorat, Mylène, Guragossian, Nathalie, Marminon, Christelle, Valdameri, Glaucio, Bollacke, Andre, Guillon, Jean, Pinaud, Noël, Marchivie, Mathieu, Cadena, Silvia M, Jose, Joachim, Le Borgne, Marc, Di Pietro, Attilio
Publicado no Drug Des Devel Ther (2015)

Azaindole derivatives are inhibitors of microtubule dynamics, with anti-cancer and anti-angiogenic activities

Por Prudent, Renaud, Vassal-Stermann, Émilie, Nguyen, Chi-Hung, Mollaret, Marjorie, Viallet, Jean, Desroches-Castan, Agnès, Martinez, Anne, Barette, Caroline, Pillet, Catherine, Valdameri, Glaucio, Soleilhac, Emmanuelle, Di Pietro, Attilio, Feige, Jean-Jacques, Billaud, Marc, Florent, Jean-Claude, Lafanechère, Laurence
Publicado em 2013

New structure–activity relationships of chalcone inhibitors of breast cancer resistance protein: polyspecificity toward inhibition and critical substitutions against cytotoxicity

Por Rangel, Luciana Pereira, Winter, Evelyn, Gauthier, Charlotte, Terreux, Raphaël, Chiaradia-Delatorre, Louise D, Mascarello, Alessandra, Nunes, Ricardo J, Yunes, Rosendo A, Creczynski-Pasa, Tania B, Macalou, Sira, Lorendeau, Doriane, Baubichon-Cortay, Hélène, Ferreira-Pereira, Antonio, Di Pietro, Attilio
Publicado em 2013

Dicer-Mediated Upregulation of BCRP Confers Tamoxifen Resistance in Human Breast Cancer Cells

Por Selever, Jennifer, Gu, Guowei, Lewis, Michael T., Beyer, Amanda, Herynk, Matthew H., Covington, Kyle R., Tsimelzon, Anna, Dontu, Gabriela, Provost, Patrick, Di Pietro, Attilio, Boumendjel, Ahcène, Albain, Kathy, Miele, Lucio, Weiss, Heidi, Barone, Ines, Ando, Sebastiano, Fuqua, Suzanne A. W.
Publicado em 2011