Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity

Ketonic indeno[1,2-b]indole-9,10-dione derivatives, initially designed as human casein kinase II (CK2) inhibitors, were recently shown to be converted into efficient inhibitors of drug efflux by the breast cancer resistance protein ABCG2 upon suited substitutions including a N(5)-phenethyl on C-ring...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Drug Des Devel Ther
Egile Nagusiak: Gozzi, Gustavo Jabor, Bouaziz, Zouhair, Winter, Evelyn, Daflon-Yunes, Nathalia, Honorat, Mylène, Guragossian, Nathalie, Marminon, Christelle, Valdameri, Glaucio, Bollacke, Andre, Guillon, Jean, Pinaud, Noël, Marchivie, Mathieu, Cadena, Silvia M, Jose, Joachim, Le Borgne, Marc, Di Pietro, Attilio
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Dove Medical Press 2015
Gaiak:
Original Research
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4498724/
https://ncbi.nlm.nih.gov/pubmed/26170632
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2147/DDDT.S84982
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