(S)-4-Trimethylsilyl-3-butyn-2-ol as an auxiliary for stereocontrolled synthesis of salinosporamide analogs with modifications at positions C2 and C5

Por Blasdel, Landy K., Lee, DongEun, Sun, Binyuan, Myers, Andrew G.
Publicado em 2013

Structure-activity relationships and docking studies of synthetic 2-arylindole derivatives determined with aromatase and quinone reductase 1

Por Prior, Allan M., Yu, Xufen, Park, Eun-Jung, Kondratyuk, Tamara P., Lin, Yan, Pezzuto, John M., Sun, Dianqing
Publicado no Bioorg Med Chem Lett (2017)

Design, synthesis, and biological evaluation of callophycin A and analogues as potential chemopreventive and anticancer agents

Por Shen, Li, Park, Eun-Jung, Kondratyuk, Tamara P., Guendisch, Daniela, Marler, Laura, Pezzuto, John M., Wright, Anthony D., Sun, Dianqing
Publicado em 2011

Synthesis and Biological Evaluation of Manassantin Analogues for Hypoxia-Inducible Factor 1α Inhibition

Por Kwon, Do-Yeon, Lee, Hye Eun, Weitzel, Douglas H., Park, Kyunghye, Lee, Sun Hee, Lee, Chen-Ting, Stephenson, Tesia N., Park, Hyeri, Fitzgerald, Michael C., Chi, Jen-Tsan, Mook, Robert A., Dewhirst, Mark W., Lee, You Mie, Hong, Jiyong
Publicado no J Med Chem (2015)

Synthesis, Optimization and Structure-Activity Relationships of 3,5-Disubstituted Isoxazolines as New Anti-tuberculosis Agents

Por Rakesh, Dianqing Sun, Lee, Robin B., Tangallapally, Rajendra, Lee, Richard E.
Publicado em 2008

New Insights into Structure–Activity Relationship of Ipomoeassin F from Its Bioisosteric 5-Oxa/Aza Analogues

Por Zong, Guanghui, Sun, Xianwei, Bhakta, Rima, Whisenhunt, Lucas, Hu, Zhijian, Wang, Feng, Shi, Wei Q.
Publicado no Eur J Med Chem (2017)

Synthesis, evaluation, and CoMFA study of fluoroquinophenoxazine derivatives as bacterial topoisomerase IA inhibitors

Por Yu, Xufen, Zhang, Mingming, Annamalai, Arasu, Bansod, Priyanka, Narula, Gagandeep, Tse-Dinh, Yuk-Ching, Sun, Dianqing
Publicado no Eur J Med Chem (2016)

2-(3-Fluoro-4-methylsulfonylaminophenyl) Propanamides as Potent Transient Receptor Potential Vanilloid 1 (TRPV1) Antagonists: Structure Activity Relationships of 2-Amino Derivative...

Por Kim, Myeong Seop, Ryu, HyungChul, Kang, Dong Wook, Cho, Seong-Hee, Seo, Sejin, Park, Young Soo, Kim, Mi-Yeon, Kwak, Eun Joo, Kim, Yong Soo, Bhondwe, Rahul S., Kim, Ho Shin, Park, Seul-gi, Son, Karam, Choi, Sun, DeAndrea-Lazarus, Ian, Pearce, Larry V., Blumberg, Peter M., Frank, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Kögel, Babette Y., Schiene, Klaus, Christoph, Thomas, Lee, Jeewoo
Publicado em 2012

Monocarbonyl analogs of curcumin inhibit growth of antibiotic sensitive and resistant strains of Mycobacterium tuberculosis

Por Baldwin, Patrick R., Reeves, Analise Z., Powell, Kimberly R., Napier, Ruth J., Swimm, Alyson I., Sun, Aiming, Giesler, Kyle, Bommarius, Bettina, Shinnick, Thomas M., Snyder, James P., Liotta, Dennis C., Kalman, Daniel
Publicado no Eur J Med Chem (2015)

Anti-inflammatory hybrids of secondary amines and amide-sulfamide derivatives

Por Bai, Renren, Sun, Jian, Liang, Zhongxing, Yoon, Younghyoun, Salgado, Eric, Feng, Amber, Oum, Yoonhyeun, Xie, Yuanyuan, Shim, Hyunsuk
Publicado no Eur J Med Chem (2018)

Synthesis and structure-activity relationship studies of novel 3,9-substituted α-carboline derivatives with high cytotoxic activity against colorectal cancer cells

Por Lin, Yi-Chien, Chen, Yi-Fong, Tseng, Li-Shin, Lee, Yueh-Hsuan, Morris-Natschke, Susan L, Kuo, Sheng-Chu, Yang, Ning-Sun, Lee, Kuo-Hsiung, Huang, Li-Jiau
Publicado no Eur J Med Chem (2016)

Hydrogen Peroxide Activated Quinone Methide Precursors with Enhanced DNA Cross-Linking Capability and Cytotoxicity towards Cancer Cells

Por Wang, Yibin, Fan, Heli, Balakrishnan, Kumudha, Lin, Zechao, Cao, Sheng, Chen, Wenbing, Fan, Yukai, Guthrie, Quibria A., Sun, Huabing, Teske, Kelly A., Gandhi, Varsha, Arnold, Leggy A., Peng, Xiaohua
Publicado no Eur J Med Chem (2017)

Synthesis and biological evaluations of chalcones, flavones and chromenes as farnesoid x receptor (FXR) antagonists

Por Zhang, Guoning, Liu, Shuainan, Tan, Wenjuan, Verma, Ruchi, Chen, Yuan, Sun, Deyang, Huan, Yi, Jiang, Qian, Wang, Xing, Wang, Na, Xu, Yang, Wong, Chiwai, Shen, Zhufang, Deng, Ruitang, Liu, Jinsong, Zhang, Yanqiao, Fang, Weishuo
Publicado no Eur J Med Chem (2017)