Pyrazole C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists

par Lee, Sunho, Kim, Changhoon, Ann, Jihyae, Thorat, Shivaji A., Kim, Eunhye, Park, Jongmi, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Publié dans Bioorg Med Chem Lett (2017)

t-Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists

par Lee, Sunho, Kang, Dong Wook, Ryu, HyungChul, Kim, Changhoon, Ann, Jihyae, Lee, Hobin, Kim, Eunhye, Hong, Sunhye, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Publié dans Bioorg Med Chem (2017)

Structure activity relationships of benzyl C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists

par Ann, Jihyae, Jung, Aeran, Kim, Mi-Yeon, Kim, Hyuk-Min, Ryu, HyungChul, Kim, Sunjoo, Kang, Dong Wook, Hong, Sunhye, Cui, Minghua, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Publié dans Bioorg Med Chem (2015)

α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists

par Tran, Phuong-Thao, Kim, Ho Shin, Ann, Jihyae, Kim, Sung-Eun, Kim, Changhoon, Hong, Mannkyu, Hoang, Van-Hai, Ngo, Van T. H., Hong, Sunhye, Cui, Minghua, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, Jeewoo
Publié dans Bioorg Med Chem Lett (2015)

Pyridine C-region analogs of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists

par Ryu, HyungChul, Seo, Sejin, Lee, Jee-Young, Ha, Tae-Hwan, Lee, Sunho, Jung, Aeran, Ann, Jihyae, Kim, Sung-Eun, Yoon, Suyoung, Hong, Mannkyu, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Schiene, Klaus, Stockhausen, Hannelore, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo
Publié dans Eur J Med Chem (2015)

2-Alkyl/alkenyl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists

par Ryu, HyungChul, Seo, Sejin, Cho, Seong-Hee, Kim, Ho Shin, Jung, Aeran, Kang, Dong Wook, Son, Karam, Cui, Minghua, Hong, Sun-hye, Sharma, Pankaz Kumar, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Schiene, Klaus, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo
Publié dans Bioorg Med Chem Lett (2014)

2-(3-Fluoro-4-methylsulfonylaminophenyl) Propanamides as Potent Transient Receptor Potential Vanilloid 1 (TRPV1) Antagonists: Structure Activity Relationships of 2-Amino Derivative...

par Kim, Myeong Seop, Ryu, HyungChul, Kang, Dong Wook, Cho, Seong-Hee, Seo, Sejin, Park, Young Soo, Kim, Mi-Yeon, Kwak, Eun Joo, Kim, Yong Soo, Bhondwe, Rahul S., Kim, Ho Shin, Park, Seul-gi, Son, Karam, Choi, Sun, DeAndrea-Lazarus, Ian, Pearce, Larry V., Blumberg, Peter M., Frank, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Kögel, Babette Y., Schiene, Klaus, Christoph, Thomas, Lee, Jeewoo
Publié 2012