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New Insights into Structure–Activity Relationship of Ipomoeassin F from Its Bioisosteric 5-Oxa/Aza Analogues

Ipomoeassin F, a plant-derived macrolide, exhibited single-digit nanomolar growth inhibition activity against many cancer cell lines. In this report, a series of 5-oxa/aza analogues was prepared and screened for cytotoxicity. Replacement of 5-CH(2) with O/NH simplified the synthesis and led to only...

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Detalhes bibliográficos
Publicado no:Eur J Med Chem
Main Authors: Zong, Guanghui, Sun, Xianwei, Bhakta, Rima, Whisenhunt, Lucas, Hu, Zhijian, Wang, Feng, Shi, Wei Q.
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5800971/
https://ncbi.nlm.nih.gov/pubmed/29291442
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2017.11.022
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