Inhibitors for the Vitamin D Receptor–Coregulator Interaction

অনুযায়ী Teske, Kelly A., Yu, Olivia, Arnold, Leggy A.
প্রকাশিত Vitam Horm (2015)

Inhibition of hedgehog signaling by stereochemically defined des-triazole itraconazole analogues

অনুযায়ী Wen, Jiachen, Teske, Kelly A., Hadden, M. Kyle
প্রকাশিত Bioorg Med Chem Lett (2019)

Novel VDR antagonists based on the GW0742 scaffold

অনুযায়ী Teske, Kelly A., Bogart, Jonathan W., Arnold, Leggy A.
প্রকাশিত Bioorg Med Chem Lett (2017)

Structure-Activity Relationships for Itraconazole-Based Triazolone Analogues as Hedgehog Pathway Inhibitors

অনুযায়ী Pace, Jennifer R., Teske, Kelly A., Chau, Lianne Q., Wechsler-Reya, Robert J., Hadden, M. Kyle
প্রকাশিত J Med Chem (2019)

Development of Posaconazole-based Analogues as Hedgehog Signaling Pathway Inhibitors

অনুযায়ী Teske, Kelly A., Dash, Radha Charan, Morel, Shana R., Chou, Lianne Q., Wechsler-Reya, Robert J., Hadden, M. Kyle
প্রকাশিত Eur J Med Chem (2018)

Probing the ligand binding pocket of BTN3A1

অনুযায়ী Poe, Michael M., Agabiti, Sherry S., Liu, Caroline, Li, Victoria, Teske, Kelly A., Christine Hsiao, Chia-Hung, Wiemer, Andrew J.
প্রকাশিত J Med Chem (2019)

A parallel chemistry approach to identify novel nuclear receptor ligands based on the GW0742 scaffold

অনুযায়ী Teske, Kelly A., Rai, Ganesha, Nandhikonda, Premchendar, Sidhu, Preetpal S., Feleke, Belaynesh, Simeonov, Anton, Yasgar, Adam, Jadhav, Ajit, Maloney, David J., Arnold, Leggy A.
প্রকাশিত ACS Comb Sci (2017)

Synthesis and Evaluation of Vitamin D Receptor-Mediated Activities of Cholesterol and Vitamin D Metabolites

অনুযায়ী Teske, Kelly A., Bogart, Jonathan W., Sanchez, Luis M., Yu, Olivia B., Preston, Joshua V., Cook, James M., Silvaggi, Nicholas R., Bikle, Daniel D., Arnold, Leggy A.
প্রকাশিত Eur J Med Chem (2016)

Hydrogen Peroxide Activated Quinone Methide Precursors with Enhanced DNA Cross-Linking Capability and Cytotoxicity towards Cancer Cells

অনুযায়ী Wang, Yibin, Fan, Heli, Balakrishnan, Kumudha, Lin, Zechao, Cao, Sheng, Chen, Wenbing, Fan, Yukai, Guthrie, Quibria A., Sun, Huabing, Teske, Kelly A., Gandhi, Varsha, Arnold, Leggy A., Peng, Xiaohua
প্রকাশিত Eur J Med Chem (2017)

Antitumor Activity of 3-Indolylmethanamines 31B and PS121912

অনুযায়ী Guthrie, Margaret L, Sidhu, Preetpal S., Hill, Emily K., Horan, Timothy C., Nandhikonda, Premchendar, Teske, Kelly A., Yuan, Nina Y., Sidorko, Marina, Kodali, Revathi, Cook, James M., Han, Lanlan, Silvaggi, Nicholas R., Bikle, Daniel D., Moore, Richard G., Singh, Rakesh K., Arnold, Leggy A.
প্রকাশিত Anticancer Res (2015)

Synthesis and characterization of a novel gamma-aminobutyric acid type A (GABA(A)) receptor ligand that combines outstanding metabolic stability, pharmacokinetics, and anxiolytic e...

অনুযায়ী Poe, Michael M., Methuku, Kashi Reddy, Li, Guanguan, Verma, Ashwini R., Teske, Kelly A., Stafford, Douglas C., Arnold, Leggy A., Cramer, Jeffrey W., Jones, Timothy M., Cerne, Rok, Krambis, Michael J., Witkin, Jeffrey M., Jambrina, Enrique, Rehman, Sabah, Ernst, Margot, Cook, James M., Schkeryantz, Jeffrey M.
প্রকাশিত J Med Chem (2016)