Rapid access to morphinones: removal of 4, 5-ether bridge with Pd-catalyzed triflate reduction

von Hupp, Christopher D., Neumeyer, John L.
Veröffentlicht 2010

High Affinity of Carbamate Analogues of Morphinan atOpioid Receptors

von Peng, Xuemei, Knapp, Brian I., M.Bidlack, Jean, Neumeyer, John L.
Veröffentlicht 2007

In-vitro Investigation of Oxazol and Urea Analogues of Morphinan at Opioid Receptors

von Peng, Xuemei, Knapp, Brian I., Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2007

Synthesis and Pharmacological Evaluation of Hydrophobic Esters and Ethers of Butorphanol at Opioid Receptors

von Fulton, Brian S., Knapp, Brian I., Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2008

Effect of Linker Substitution on the Binding of Butorphan Univalent and Bivalent Ligands to Opioid Receptors

von Fulton, Brian S., Knapp, Brian L., Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2010

Pharmacological Properties of Bivalent Ligands Containing Butorphan Linked to Nalbuphine, Naltrexone and Naloxone at μ, δ and κ Opioid Receptors

von Peng, Xuemei, Knapp, Brian I., Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2007

Behavioral effects of the R-(+)- and S-(−) enantiomers of the D(1)-like partial receptor agonist SKF 83959 in monkeys

von Desai, Rajeev I., Neumeyer, John L., Paronis, Carol A., Nguyen, Phong, Bergman, Jack
Veröffentlicht 2006

In Vivo Characterization of (−)(−)MCL-144 and (+)(−)MCL-193: Isomeric, Bivalent Ligands with Mu/Kappa Agonist Properties

von Mathews, Jennifer L., Fulton, Brian S., Negus, S. Stevens, Neumeyer, John L., Bidlack, Jean M.
Veröffentlicht 2008

Synthesis and Opioid Receptor Binding Affinities of 2-Substituted and 3-Aminomorphinans: Ligands for mu, kappa and delta Opioid Receptors

von Decker, Michael, Si, Yu-Gui, Knapp, Brian I., Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2010

Univalent and Bivalent Ligands of Butorphan: Characteristics of the Linking Chain determine the Affinity and Potency of Such Opioid Ligands

von Decker, Michael, Fulton, Brian S., Zhang, Bin, Knapp, Brian I., Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2009

Synthesis and Binding Affinity of Novel Mono- and Bivalent Morphinan Ligands for κ, μ and δ Opioid Receptors

von Zhang, Bin, Zhang, Tangzhi, Sromek, Anna W., Scrimale, Thomas, Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2011

Synthesis and Evaluation of Fluorinated Aporphines: Potential Positron Emission Tomography Ligands for D(2) Receptors

von Sromek, Anna W., Si, Yu-Gui, Zhang, Tangzhi, George, Susan R., Seeman, Philip, Neumeyer, John L.
Veröffentlicht 2011

Aminothiazolomorphinans with Mixed Kappa and Mu Opioid Activity

von Zhang, Tangzhi, Yan, Zhaohua, Sromek, Anna, Knapp, Brian I., Scrimale, Thomas, Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2011

Arylbenzazepines Are Potent Modulators for the Delayed Rectifier K(+) Channel: A Potential Mechanism for Their Neuroprotective Effects

von Chen, Xue-Qin, Zhang, Jing, Neumeyer, John L., Jin, Guo-Zhang, Hu, Guo-Yuan, Zhang, Ao, Zhen, Xuechu
Veröffentlicht 2009

Synthesis, Binding Affinity, and Functional In Vitro Activity of 3-Benzylaminomorphinan and 3-Benzylaminomorphine Ligands at Opioid Receptors

von Neumeyer, John L., Zhang, Bin, Zhang, Tangzhi, Sromek, Anna W., Knapp, Brian I., Cohen, Dana J., Bidlack, Jean M.
Veröffentlicht 2012

Preliminary Pharmacological Evaluation of Enantiomeric Morphinans

von Sromek, Anna W., Provencher, Brian A., Russell, Shayla, Chartoff, Elena, Knapp, Brian I., Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2014

New Opioid Designed Multiple Ligand from Dmt-Tic and Morphinan Pharmacophores

von Neumeyer, John L., Peng, Xuemei, Knapp, Brian I., Bidlack, Jean M., Lazarus, Lawrence H., Salvadori, Severo, Trapella, Claudio, Balboni, Gianfranco
Veröffentlicht 2006

Evolution of the Bifunctional Lead μ Agonist/δ Antagonist Containing the 2′,6′-Dimethyl-l-tyrosine−1,2,3,4-Tetrahydroisoquinoline-3-carboxylic Acid (Dmt−Tic) Opioid Pharmacophore...

von Balboni, Gianfranco, Salvadori, Severo, Trapella, Claudio, Knapp, Brian I., Bidlack, Jean M., Lazarus, Lawrence H., Peng, Xuemei, Neumeyer, John L.
Veröffentlicht 2009

Synthesis and Pharmacological Evaluation Aminothiazolomorphinans at Mu and Kappa Opioid Receptors

von Provencher, Brian A., Sromek, Anna W., Li, Wei, Russell, Shayla, Chartoff, Elena, Knapp, Brian I., Bidlack, Jean M., Neumeyer, John L.
Veröffentlicht 2013

Opioid Bifunctional Ligands from Morphine and the Opioid Pharmacophore Dmt-Tic

von Balboni, Gianfranco, Salvadori, Severo, Marczak, Ewa D., Knapp, Brian I., Bidlack, Jean M., Lazarus, Lawrence H., Peng, Xuemei, Si, Yu Gui, Neumeyer, John L.
Veröffentlicht 2010