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Synthesis and Binding Affinity of Novel Mono- and Bivalent Morphinan Ligands for κ, μ and δ Opioid Receptors

A novel series of homo- and heterodimeric ligands containing κ/μ agonist and μ agonist/antagonist pharmacophores joined by a 10-carbon ester linker chain were synthesized and evaluated for their in vitro binding affinity at κ, μ, and δ opioid receptors and their functional activities were determined...

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Autori principali: Zhang, Bin, Zhang, Tangzhi, Sromek, Anna W., Scrimale, Thomas, Bidlack, Jean M., Neumeyer, John L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3095849/
https://ncbi.nlm.nih.gov/pubmed/21482470
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2011.03.052
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