Synthesis and SAR of Thiazolylmethylphenyl Glucoside as Novel C-Aryl Glucoside SGLT2 Inhibitors

Por Song, Kwang-Seop, Lee, Suk Ho, Kim, Min Ju, Seo, Hee Jeong, Lee, Junwon, Lee, Sung-Han, Jung, Myung Eun, Son, Eun-Jung, Lee, MinWoo, Kim, Jeongmin, Lee, Jinhwa
Publicado em 2010

Use of Ionically Tagged Glycosyl Donors in the Synthesis of Oligosaccharide Libraries

Por Kim, Eun Ju, Gray, Gary R.
Publicado em 2009

Tat-DJ-1 inhibits oxidative stress-mediated RINm5F cell death through suppression of NF-κB and MAPK activation

Por Jo, Hyo Sang, Cha, Hyun Ju, Kim, Sang Jin, Yeo, Hyeon Ji, Cho, Su Bin, Park, Jung Hwan, Lee, Chi Hern, Yeo, Eun Ji, Choi, Yeon Joo, Eum, Won Sik, Choi, Soo Young
Publicado no Med Chem Res (2016)

Non-proteinogenic amino acids in the pThr-2 position of a pentamer peptide that confer high binding affinity for the polo box domain (PBD) of polo-like kinase 1 (Plk1)

Por Qian, Wen-Jian, Park, Jung-Eun, Lee, Kyung S., Burke, Terrence R.
Publicado em 2012

Effects on Polo-like Kinase 1 Polo-box Domain Binding Affinities of Peptides Incurred by Structural Variation at the Phosphoamino Acid Position

Por Qian, Wenjian, Park, Jung-Eun, Liu, Fa, Lee, Kyung S., Burke, Terrence R.
Publicado em 2012

Probing Binding Modes of Small Molecule Inhibitors to the Polo-Box Domain of Human Polo-like Kinase 1

Por Liao, Chenzhong, Park, Jung-Eun, Bang, Jeong K., Nicklaus, Marc C., Lee, Kyung S.
Publicado em 2010

Effect of cinnamamides on atopic dermatitis through regulation of IL-4 in CD4(+) cells

Por Choi, Eun-Ju, Ryu, Young Bae, Tang, Yujiao, Kim, Bo Ram, Lee, Woo Song, Debnath, Trishna, Fan, Meiqi, Kim, Eun-Kyung, Lee, Hyun-Su
Publicado no J Enzyme Inhib Med Chem (2019)

Optimizing Thiadiazole Analogues of Resveratrol vs. Three Chemopreventive Targets

Por Mayhoub, Abdelrahman S., Marler, Laura, Kondratyuk, Tamara, Park, Eun-Jung, Pezzuto, John M., Cushman, Mark
Publicado em 2011

Optimization of Thiazole Analogues of Resveratrol for Induction of NAD(P)H:quinone Reductase 1 (QR1)

Por Mayhoub, Abdelrahman S., Marler, Laura, Kondratyuk, Tamara P., Park, Eun-Jung, Pezzuto, John M., Cushman, Mark
Publicado em 2012

Epimeric methylsulfinyladenosine derivatives from the marine ascidian Herdmania momus

Por Li, Jian Lin, Kim, Eun La, Wang, Haibo, Hong, Jongki, Shin, Sook, Lee, Chong-Kyo, Jung, Jee H.
Publicado no Bioorg Med Chem Lett (2013)

Structure-activity relationships and docking studies of synthetic 2-arylindole derivatives determined with aromatase and quinone reductase 1

Por Prior, Allan M., Yu, Xufen, Park, Eun-Jung, Kondratyuk, Tamara P., Lin, Yan, Pezzuto, John M., Sun, Dianqing
Publicado no Bioorg Med Chem Lett (2017)

Design, synthesis, and biological evaluation of callophycin A and analogues as potential chemopreventive and anticancer agents

Por Shen, Li, Park, Eun-Jung, Kondratyuk, Tamara P., Guendisch, Daniela, Marler, Laura, Pezzuto, John M., Wright, Anthony D., Sun, Dianqing
Publicado em 2011

OGA inhibition by GlcNAc-selenazoline

Por Kim, Eun Ju, Love, Dona C., Darout, Etzer, Abdo, Mohannad, Rempel, Brian, Withers, Stephen G., Rablen, Paul R., Hanover, John A., Knapp, Spencer
Publicado em 2010

Selective Synthesis and Biological Evaluation of Sulfate-Conjugated Resveratrol Metabolites

Por Hoshino, Juma, Park, Eun-Jung, Kondratyuk, Tamara P., Marler, Laura, Pezzuto, John M., van Breemen, Richard B., Mo, Shunyan, Li, Yongchao, Cushman, Mark
Publicado em 2010

Potential Chemopreventive Agents Based on the Structure of the Lead Compound 2-Bromo-1-hydroxyphenazine, Isolated from Streptomyces sp., Strain CNS284

Por Conda-Sheridan, Martin, Marler, Laura, Park, Eun-Jung, Kondratyuk, Tamara P., Jermihov, Katherine, Mesecar, Andrew D., Pezzuto, John M., Asolkar, Ratnakar N., Fenical, William, Cushman, Mark
Publicado em 2010

Identification, Synthesis, and Biological Evaluation of the Metabolites of 3-Amino-6-(3'-aminopropyl)-5H-indeno[1,2-c]isoquinoline-5,11-(6H)dione (AM6-36), a Promising Rexinoid Lea...

Por Chen, Lian, Conda-Sheridan, Martin, Narasimha Reddy, P. V., Morrell, Andrew, Park, Eun-Jung, Kondratyuk, Tamara P., Pezzuto, John M., van Breemen, Richard B., Cushman, Mark
Publicado em 2012

Identification of a New Heterocyclic Scaffold for Inhibitors of the Polo-Box Domain of Polo-like Kinase 1

Por Alverez, Celeste N., Park, Jung-Eun, Toti, Kiran S., Xia, Yangliu, Krausz, Kristopher W., Rai, Ganesha, Bang, Jeong K., Gonzalez, Frank J., Jacobson, Kenneth A., Lee, Kyung S.
Publicado no J Med Chem (2020)

Identification of 6′-β-fluoro-homoaristeromycin as a potent inhibitor of chikungunya virus replication

Por Shin, Young Sup, Jarhad, Dnyandev B., Jang, Min Hwan, Kovacikova, Kristina, Kim, Gyudong, Yoon, Ji-seong, Kim, Hong-Rae, Hyun, Young Eum, Tipnis, Amol S., Chang, Tong-Shin, van Hemert, Martijn J., Jeong, Lak Shin
Publicado no Eur J Med Chem (2020)

Design, synthesis and biological evaluation of 2-aminoquinazolin-4(3H)-one derivatives as potential SARS-CoV-2 and MERS-CoV treatments

Por Lee, Jun Young, Shin, Young Sup, Jeon, Sangeun, Lee, Se In, Noh, Soojin, Cho, Jung-Eun, Jang, Min Seong, Kim, Seungtaek, Song, Jong Hwan, Kim, Hyoung Rae, Park, Chul Min
Publicado no Bioorg Med Chem Lett (2021)

A POTENT AND SELECTIVE INHIBITOR TARGETING HUMAN AND MURINE 12/15-LOX

Por Armstrong, Michelle M., Freedman, Cody J., Jung, Joo Eun, Zheng, Yi, Kalyanaraman, Chakrapani, Jacobson, Matthew P., Simeonov, Anton, Maloney, David J., van Leyen, Klaus, Jadhav, Ajit, Holman, Theodore R.
Publicado no Bioorg Med Chem (2016)