Efficient diastereoselective synthesis of a new class of azanucleosides: 2′-homoazanucleosides

di Bouton, Jakob, Van Hecke, Kristof, Van Calenbergh, Serge
Pubblicato in Tetrahedron (2017)

Synthesis of pyrrolidine-based hamamelitannin analogues as quorum sensing inhibitors in Staphylococcus aureus

di Bouton, Jakob, Van Hecke, Kristof, Rasooly, Reuven, Van Calenbergh, Serge
Pubblicato in Beilstein J Org Chem (2018)

Acyloxybenzyl and Alkoxyalkyl Prodrugs of a Fosmidomycin Surrogate as Antimalarial and Antitubercular Agents

di Courtens, Charlotte, Risseeuw, Martijn, Caljon, Guy, Cos, Paul, Van Calenbergh, Serge
Pubblicato in ACS Med Chem Lett (2018)

Structural basis of NKT cell inhibition using the T-cell receptor-blocking anti-CD1d antibody 1B1

di Ying, Ge, Wang, Jing, Mallevaey, Thierry, Van Calenbergh, Serge, Zajonc, Dirk M.
Pubblicato in J Biol Chem (2019)

Exploring the purine core of 3′-C-ethynyladenosine (EAdo) in search of novel nucleoside therapeutics

di Hulpia, Fabian, Balzarini, Jan, Schols, Dominique, Andrei, Graciela, Snoeck, Robert, Van Calenbergh, Serge
Pubblicato in Bioorg Med Chem Lett (2016)

Exploring human adenosine A(3) receptor complementarity and activity for adenosine analogues modified in the ribose and purine moiety

di Van Rompaey, Philippe, Jacobson, Kenneth A., Gross, Ariel S., Gao, Zhan-Guo, Van Calenbergh, Serge
Pubblicazione 2005

Synthesis of C-5″ and C-6″-modified α-GalCer analogues as iNKT-cell agonists

di Guillaume, Joren, Pauwels, Nora, Aspeslagh, Sandrine, Zajonc, Dirk M., Elewaut, Dirk, Van Calenbergh, Serge
Pubblicato in Bioorg Med Chem (2015)

Cinnamaldehyde and cinnamaldehyde derivatives reduce virulence in Vibrio spp. by decreasing the DNA-binding activity of the quorum sensing response regulator LuxR

di Brackman, Gilles, Defoirdt, Tom, Miyamoto, Carol, Bossier, Peter, Van Calenbergh, Serge, Nelis, Hans, Coenye, Tom
Pubblicazione 2008

Crystal Structures of Bovine CD1d Reveal Altered αGalCer Presentation and a Restricted A’ Pocket Unable to Bind Long-Chain Glycolipids

di Wang, Jing, Guillaume, Joren, Pauwels, Nora, Van Calenbergh, Serge, Van Rhijn, Ildiko, Zajonc, Dirk M.
Pubblicazione 2012

Synthesis and Evaluation of N(6)-Substituted Apioadenosines as Potential Adenosine A(3) Receptor Modulators

di Toti, Kiran S., Moss, Steven M., Paoletta, Silvia, Gao, Zhan-Guo, Jacobson, Kenneth A., Van Calenbergh, Serge
Pubblicazione 2014

Synthesis and structure-activity relationships of cerebroside analogues as substrates of cerebroside sulphotransferase and discovery of a competitive inhibitor

di Li, Wenjin, Guillaume, Joren, Baqi, Younis, Wachsmann, Isabell, Gieselmann, Volkmar, Van Calenbergh, Serge, Müller, Christa E.
Pubblicato in J Enzyme Inhib Med Chem (2020)

Novel Potentiators for Vancomycin in the Treatment of Biofilm-Related MRSA Infections via a Mix and Match Approach

di Vermote, Arno, Brackman, Gilles, Risseeuw, Martijn D. P., Cappoen, Davie, Cos, Paul, Coenye, Tom, Van Calenbergh, Serge
Pubblicato in ACS Med Chem Lett (2016)

Synthesis of a 3′-C-ethynyl-β-d-ribofuranose purine nucleoside library: Discovery of C7-deazapurine analogs as potent antiproliferative nucleosides

di Hulpia, Fabian, Noppen, Sam, Schols, Dominique, Andrei, Graciela, Snoeck, Robert, Liekens, Sandra, Vervaeke, Peter, Van Calenbergh, Serge
Pubblicato in Eur J Med Chem (2018)

Synthesis and P2Y Receptor Activity of Nucleoside 5′-Phosphonate Derivatives

di Cosyn, Liesbet, Van Calenbergh, Serge, Joshi, Bhalchandra V., Ko, Hyojin, Carter, Rhonda L., Harden, T. Kendall, Jacobson, Kenneth A.
Pubblicazione 2009

Synthesis and Evaluation of Amino-Modified α-GalCer Analogues

di Trappeniers, Matthias, Chofor, René, Aspeslagh, Sandrine, Li, Yali, Linclau, Bruno, Zajonc, Dirk M., Elewaut, Dirk, Van Calenbergh, Serge
Pubblicazione 2010

Structure-Activity Relationship of Cinnamaldehyde Analogs as Inhibitors of AI-2 Based Quorum Sensing and Their Effect on Virulence of Vibrio spp

di Brackman, Gilles, Celen, Shari, Hillaert, Ulrik, Van Calenbergh, Serge, Cos, Paul, Maes, Louis, Nelis, Hans J., Coenye, Tom
Pubblicazione 2011

Design, Synthesis and Characterization of a New Series of Fluorescent Metabotropic Glutamate Receptor Type 5 Negative Allosteric Modulators

di Fernández-Dueñas, Víctor, Qian, Mingcheng, Argerich, Josep, Amaral, Carolina, Risseeuw, Martijn D.P., Van Calenbergh, Serge, Ciruela, Francisco
Pubblicato in Molecules (2020)

The Quorum Sensing Inhibitor Hamamelitannin Increases Antibiotic Susceptibility of Staphylococcus aureus Biofilms by Affecting Peptidoglycan Biosynthesis and eDNA Release

di Brackman, Gilles, Breyne, Koen, De Rycke, Riet, Vermote, Arno, Van Nieuwerburgh, Filip, Meyer, Evelyne, Van Calenbergh, Serge, Coenye, Tom
Pubblicato in Sci Rep (2016)

2-Triazole-Substituted Adenosines: A New Class of Selective A(3) Adenosine Receptor Agonists, Partial Agonists, and Antagonists

di Cosyn, Liesbet, Palaniappan, Krishnan K., Kim, Soo-Kyung, Duong, Heng T., Gao, Zhan-Guo, Jacobson, Kenneth A., Van Calenbergh, Serge
Pubblicato in J Med Chem (2006)

Synthesis of Extended Uridine Phosphonates Derived from an Allosteric P2Y(2) Receptor Ligand

di Song, Lijun, Risseeuw, Martijn D. P., Karalic, Izet, Barrett, Matthew O., Brown, Kyle A., Harden, T. Kendall, Van Calenbergh, Serge
Pubblicato in Molecules (2014)