Parameterization of aromatic azido group: Application for Photoaffinity Probe in Molecular Dynamics Studies

بواسطة Pieffet, Gilles, Petukhov, Pavel A.
منشور في 2009

A One-Pot Selective Synthesis of N-Boc Protected Secondary Amines: Tandem Direct Reductive Amination/N-Boc Protection

بواسطة Neelarapu, Raghupathi, Petukhov, Pavel A.
منشور في 2012

Insights from Comprehensive Multiple Receptor Docking to HDAC8

بواسطة Brunsteiner, Michael, Petukhov, Pavel A.
منشور في 2012

Identification of Hepatitis C Virus Inhibitors Targeting Different Aspects of Infection Using a Cell-Based Assay

بواسطة Yu, Xuemei, Sainz, Bruno, Petukhov, Pavel A., Uprichard, Susan L.
منشور في 2012

Divergent JNK Phosphorylation of HDAC3 in Triple Negative Breast Cancer Cells Determines HDAC Inhibitor Binding and Selectivity

بواسطة Hanigan, Thomas W., Aboukhatwa, Shaimaa M., Taha, Taha, Frasor, Jonna, Petukhov, Pavel A.
الحاوية / القاعدة Cell Chem Biol (2017)

Scaffold dependent histone deacetylase (HDAC) inhibitor induced re-equilibration of the subcellular localization and post-translational modification state of class I HDACs

بواسطة Hanigan, Thomas W., Taha, Taha Y., Aboukhatwa, Shaimaa M., Frasor, Jonna, Petukhov, Pavel A.
الحاوية / القاعدة PLoS One (2017)

Histone deacetylase inhibitor-based chromatin precipitation for identification of targeted genomic loci

بواسطة Hanigan, Thomas W., Danes, Jeanne M., Taha, Taha Y., Frasor, Jonna, Petukhov, Pavel A.
الحاوية / القاعدة J Biol Methods (2018)

Modulation of hepatitis B virus pregenomic RNA stability and splicing by histone deacetylase 5 enhances viral biosynthesis

بواسطة Taha, Taha Y., Anirudhan, Varada, Limothai, Umaporn, Loeb, Daniel D., Petukhov, Pavel A., McLachlan, Alan
الحاوية / القاعدة PLoS Pathog (2020)

Design, Synthesis, Docking, and Biological Evaluation of Novel Diazide-containing Isoxazole- and Pyrazole-based Histone Deacetylase Probes

بواسطة Neelarapu, Raghupathi, Holzle, Denise L., Velaparthi, Subash, Bai, He, Brunsteiner, Michael, Blond, Sylvie Y., Petukhov, Pavel A.
منشور في 2011

Design, synthesis, modeling, biological evaluation and photoaffinity labeling studies of novel series of photoreactive benzamide probes for histone deacetylase 2

بواسطة Vaidya, Aditya Sudheer, Karumudi, Bhargava, Mendonca, Emma, Madriaga, Antonett, Abdelkarim, Hazem, van Breemen, Richard B., Petukhov, Pavel A.
منشور في 2012

A Chimeric SERM-Histone Deacetylase Inhibitor Approach to Breast Cancer Therapy

بواسطة Patel, Hitisha K., Siklos, Marton I., Abdelkarim, Hazem, Mendonca, Emma L., Vaidya, Aditya, Petukhov, Pavel A., Thatcher, Gregory R. J.
منشور في 2013

Kaempferol Exhibits Progestogenic Effects in Ovariectomized Rats

بواسطة Toh, May Fern, Mendonca, Emma, Eddie, Sharon L., Endsley, Michael P., Lantvit, Daniel D., Petukhov, Pavel A., Burdette, Joanna E.
الحاوية / القاعدة J Steroids Horm Sci (2014)

2-Arylidene Hydrazinecarbodithioates as Potent, Selective Inhibitors of Cystathionine γ-Lyase (CSE)

بواسطة Bhattacharjee, Abir, Sinha, Antara, Ratia, Kiira, Yin, Liang, Delgado-Rivera, Loruhama, Petukhov, Pavel A, Thatcher, Gregory R. J., Wardrop, Duncan J.
الحاوية / القاعدة ACS Med Chem Lett (2017)

Photoreactive “Nanorulers” Detect a Novel Conformation of Full length HDAC3-SMRT Complex in Solution

بواسطة Abdelkarim, Hazem, Brunsteiner, Michael, Neelarapu, Raghupathi, Bai, He, Madriaga, Antonett, van Breemen, Richard B., Blond, Sylvie Y., Gaponenko, Vadim, Petukhov, Pavel A.
منشور في 2013

Novel histone deacetylase 8 ligands without a zinc chelating group: exploring an “upside-down” binding pose

بواسطة Vaidya, Aditya Sudheer, Neelarapu, Raghupathi, Madriaga, Antonett, Bai, He, Mendonca, Emma, Abdelkarim, Hazem, van Breemen, Richard B., Blond, Sylvie Y., Petukhov, Pavel A.
منشور في 2012

Binding Ensemble PROfiling with (F)photoaffinity Labeling (BEProFL) Approach: Mapping the Binding Poses of HDAC8 Inhibitors

بواسطة He, Bai, Velaparthi, Subash, Pieffet, Gilles, Pennington, Chris, Mahesh, Aruna, Holzle, Denise L., Brunsteiner, Michael, van Breemen, Richard, Blond, Sylvie Y., Petukhov, Pavel A.
منشور في 2009

Design, Synthesis, Molecular Modeling, and Biological Evaluation of Novel Amine-based Histone Deacetylase Inhibitors

بواسطة Abdelkarim, Hazem, Neelarapu, Raghupathi, Madriaga, Antonett, Vaidya, Aditya S., Kastrati, Irida, Wang, Yue-ting, Taha, Taha Y., Thatcher, Gregory R. J., Frasor, Jonna, Petukhov, Pavel A.
الحاوية / القاعدة ChemMedChem (2017)

Platelet Protein Disulfide Isomerase Promotes Glycoprotein Ibα-Mediated Platelet-Neutrophil Interactions Under Thromboinflammatory Conditions

بواسطة Li, Jing, Kim, Kyungho, Jeong, Si-Yeon, Chiu, Joyce, Xiong, Bei, Petukhov, Pavel A., Dai, Xiangrong, Li, Xiaoyi, Andrews, Robert K., Du, Xiaoping, Hogg, Philip J., Cho, Jaehyung
الحاوية / القاعدة Circulation (2019)

Design, Synthesis, and Biological Evaluation of Tetrahydroisoquinoline-Based Histone Deacetylase 8 Selective Inhibitors

بواسطة Taha, Taha Y., Aboukhatwa, Shaimaa M., Knopp, Rachel C., Ikegaki, Naohiko, Abdelkarim, Hazem, Neerasa, Jayaprakash, Lu, Yunlong, Neelarapu, Raghupathi, Hanigan, Thomas W., Thatcher, Gregory R. J., Petukhov, Pavel A.
الحاوية / القاعدة ACS Med Chem Lett (2017)

Correction to Design, Synthesis, and Biological Evaluation of Tetrahydroisoquinoline-Based Histone Deacetylase 8 Selective Inhibitors

بواسطة Taha, Taha Y., Aboukhatwa, Shaimaa M., Knopp, Rachel C., Ikegaki, Naohiko, Abdelkarim, Hazem, Neerasa, Jayaprakash, Lu, Yunlong, Neelarapu, Raghupathi, Hanigan, Thomas W., Thatcher, Gregory R. J., Petukhov, Pavel A.
الحاوية / القاعدة ACS Med Chem Lett (2019)