Insights from Selective Non-phosphinic Inhibitors of MMP-12 Tailored to Fit with an S(1)′ Loop Canonical Conformation

por Devel, Laurent, Garcia, Sandra, Czarny, Bertrand, Beau, Fabrice, Lajeunesse, Evelyne, Vera, Laura, Georgiadis, Dimitris, Stura, Enrico, Dive, Vincent
Publicado 2010

Novel mechanism of inhibition of human angiotensin-I-converting enzyme (ACE) by a highly specific phosphinic tripeptide

por Akif, Mohd, Schwager, Sylva L., Anthony, Colin S., Czarny, Bertrand, Beau, Fabrice, Dive, Vincent, Sturrock, Edward D., Acharya, K. Ravi
Publicado 2011

Molecular Determinants of Matrix Metalloproteinase-12 Covalent Modification by a Photoaffinity Probe: INSIGHTS INTO ACTIVITY-BASED PROBE DEVELOPMENT AND CONFORMATIONAL VARIABILIT...

por Dabert-Gay, Anne-Sophie, Czarny, Bertrand, Devel, Laurent, Beau, Fabrice, Lajeunesse, Evelyne, Bregant, Sarah, Thai, Robert, Yiotakis, Athanasios, Dive, Vincent
Publicado 2008

Simple Pseudo-dipeptides with a P(2)′ Glutamate: A NOVEL INHIBITOR FAMILY OF MATRIX METALLOPROTEASES AND OTHER METZINCINS

por Devel, Laurent, Beau, Fabrice, Amoura, Mehdi, Vera, Laura, Cassar-Lajeunesse, Evelyne, Garcia, Sandra, Czarny, Bertrand, Stura, Enrico A., Dive, Vincent
Publicado 2012

Biodistribution of Nanostructured Lipid Carriers in Mice Atherosclerotic Model

por Devel, Laurent, Almer, Gunter, Cabella, Claudia, Beau, Fabrice, Bernes, Mylène, Oliva, Paolo, Navarro, Fabrice, Prassl, Ruth, Mangge, Harald, Texier, Isabelle
Publicado en Molecules (2019)

Inhibitors of BMP‐1/tolloid‐like proteinases: efficacy, selectivity and cellular toxicity

por Talantikite, Maya, Lécorché, Pascaline, Beau, Fabrice, Damour, Odile, Becker‐Pauly, Christoph, Ho, Wen‐Bin, Dive, Vincent, Vadon‐Le Goff, Sandrine, Moali, Catherine
Publicado en FEBS Open Bio (2018)

Crystal structures of highly specific phosphinic tripeptide enantiomers in complex with the angiotensin‐I converting enzyme

por Masuyer, Geoffrey, Akif, Mohd, Czarny, Bertrand, Beau, Fabrice, Schwager, Sylva L. U., Sturrock, Edward D., Isaac, R. Elwyn, Dive, Vincent, Acharya, K. Ravi
Publicado 2013

A Selective Matrix Metalloproteinase-12 Inhibitor Retards Atherosclerotic Plaque Development in Apolipoprotein E–Knockout Mice

por Johnson, Jason L., Devel, Laurent, Czarny, Bertrand, George, Sarah J., Jackson, Christopher L., Rogakos, Vassilis, Beau, Fabrice, Yiotakis, Athanasios, Newby, Andrew C., Dive, Vincent
Publicado 2011

Structural Framework for Covalent Inhibition of Clostridium botulinum Neurotoxin A by Targeting Cys(165)

por Stura, Enrico A., Le Roux, Laura, Guitot, Karine, Garcia, Sandra, Bregant, Sarah, Beau, Fabrice, Vera, Laura, Collet, Guillaume, Ptchelkine, Denis, Bakirci, Huseyin, Dive, Vincent
Publicado 2012

Optical imaging of MMP-12 active form in inflammation and aneurysm

por Razavian, Mahmoud, Bordenave, Thomas, Georgiadis, Dimitris, Beau, Fabrice, Zhang, Jiasheng, Golestani, Reza, Toczek, Jakub, Jung, Jae-Joon, Ye, Yunpeng, Kim, Hye-Yeong, Han, Jinah, Dive, Vincent, Devel, Laurent, Sadeghi, Mehran M.
Publicado en Sci Rep (2016)

Novel Matrix Metalloproteinase 12 selective radiotracers for vascular molecular imaging

por Toczek, Jakub, Bordenave, Thomas, Gona, Kiran, Kim, Hye-Yeong, Beau, Fabrice, Georgiadis, Dimitris, Correia, Isabelle, Ye, Yunpeng, Razavian, Mahmoud, Jung, Jae-Joon, Lequin, Olivier, Dive, Vincent, Sadeghi, Mehran M., Devel, Laurent
Publicado en J Med Chem (2019)

High throughput screening identifies disulfide isomerase DsbC as a very efficient partner for recombinant expression of small disulfide-rich proteins in E. coli

por Nozach, Hervé, Fruchart-Gaillard, Carole, Fenaille, François, Beau, Fabrice, Ramos, Oscar Henrique Pereira, Douzi, Badreddine, Saez, Natalie J, Moutiez, Mireille, Servent, Denis, Gondry, Muriel, Thaï, Robert, Cuniasse, Philippe, Vincentelli, Renaud, Dive, Vincent
Publicado 2013

Synthesis, in vitro and in vivo evaluation of MMP-12 selective optical probes

por Bordenave, Thomas, Helle, Marion, Beau, Fabrice, Georgiadis, Dimitris, Tepshi, Livia, Bernes, Mylène, Ye, Yunpeng, Levenez, Laure, Poquet, Enora, Nozach, Hervé, Razavian, Mahmoud, Toczek, Jakub, Stura, Enrico A., Dive, Vincent, Sadeghi, Mehran M., Devel, Laurent
Publicado en Bioconjug Chem (2016)

Green mamba peptide targets type-2 vasopressin receptor against polycystic kidney disease

por Ciolek, Justyna, Reinfrank, Helen, Quinton, Loïc, Viengchareun, Say, Stura, Enrico A., Vera, Laura, Sigismeau, Sabrina, Mouillac, Bernard, Orcel, Hélène, Peigneur, Steve, Tytgat, Jan, Droctové, Laura, Beau, Fabrice, Nevoux, Jerome, Lombès, Marc, Mourier, Gilles, De Pauw, Edwin, Servent, Denis, Mendre, Christiane, Witzgall, Ralph, Gilles, Nicolas
Publicado en Proc Natl Acad Sci U S A (2017)