Self-cleavage of the Pseudomonas aeruginosa Cell-surface Signaling Anti-sigma Factor FoxR Occurs through an N-O Acyl Rearrangement

di Bastiaansen, Karlijn C., van Ulsen, Peter, Wijtmans, Maikel, Bitter, Wilbert, Llamas, María A.
Pubblicato in J Biol Chem (2015)

Metabolic profiling of ligands for the chemokine receptor CXCR3 by liquid chromatography-mass spectrometry coupled to bioaffinity assessment

di Mladic, Marija, Scholten, Danny J., Wijtmans, Maikel, Falck, David, Leurs, Rob, Niessen, Wilfried M. A., Smit, Martine J., Kool, Jeroen
Pubblicato in Anal Bioanal Chem (2015)

Targeted LC–MS derivatization for aldehydes and carboxylic acids with a new derivatization agent 4-APEBA

di Eggink, Mark, Wijtmans, Maikel, Kretschmer, Ansgar, Kool, Jeroen, Lingeman, Henk, de Esch, Iwan J. P., Niessen, Wilfried M. A., Irth, Hubertus
Pubblicazione 2010

Exploring the Effect of Cyclization of Histamine H(1) Receptor Antagonists on Ligand Binding Kinetics

di Wang, Zhiyong, Bosma, Reggie, Kuhne, Sebastiaan, van den Bor, Jelle, Garabitian, Wrej, Vischer, Henry F., Wijtmans, Maikel, Leurs, Rob, de Esch, Iwan J.P.
Pubblicato in ACS Omega (2021)

Bromo-Cyclobutenaminones as New Covalent UDP-N-Acetylglucosamine Enolpyruvyl Transferase (MurA) Inhibitors

di Hamilton, David J., Ábrányi-Balogh, Péter, Keeley, Aaron, Petri, László, Hrast, Martina, Imre, Tímea, Wijtmans, Maikel, Gobec, Stanislav, de Esch, Iwan J. P., Keserű, György Miklós
Pubblicato in Pharmaceuticals (Basel) (2020)

A Photoswitchable Agonist for the Histamine H(3) Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor

di Hauwert, Niels J., Mocking, Tamara A. M., Da Costa Pereira, Daniel, Lion, Ken, Huppelschoten, Yara, Vischer, Henry F., De Esch, Iwan J. P., Wijtmans, Maikel, Leurs, Rob
Pubblicato in Angew Chem Int Ed Engl (2019)

Covalent Inhibition of the Histamine H(3) Receptor

di Wágner, Gábor, Mocking, Tamara A. M., Kooistra, Albert J., Slynko, Inna, Ábrányi-Balogh, Péter, Keserű, György M., Wijtmans, Maikel, Vischer, Henry F., de Esch, Iwan J. P., Leurs, Rob
Pubblicato in Molecules (2019)

Combined CXCR3/CXCR4 measurements are of high prognostic value in chronic lymphocytic leukemia due to negative co-operativity of the receptors

di Ganghammer, Sylvia, Gutjahr, Julia, Hutterer, Evelyn, Krenn, Peter W., Pucher, Susanne, Zelle-Rieser, Claudia, Jöhrer, Karin, Wijtmans, Maikel, Leurs, Rob, Smit, Martine J., Gattei, Valter, Greil, Richard, Hartmann, Tanja N.
Pubblicato in Haematologica (2016)

A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light

di Gómez-Santacana, Xavier, de Munnik, Sabrina M, Mocking, Tamara A M, Hauwert, Niels J, Sun, Shanliang, Vijayachandran, Prashanna, de Esch, Iwan J P, Vischer, Henry F, Wijtmans, Maikel, Leurs, Rob
Pubblicato in Beilstein J Org Chem (2019)

Route to Prolonged Residence Time at the Histamine H(1) Receptor: Growing from Desloratadine to Rupatadine

di Bosma, Reggie, Wang, Zhiyong, Kooistra, Albert J., Bushby, Nick, Kuhne, Sebastiaan, van den Bor, Jelle, Waring, Michael J., de Graaf, Chris, de Esch, Iwan J., Vischer, Henry F., Sheppard, Robert J., Wijtmans, Maikel, Leurs, Rob
Pubblicato in J Med Chem (2019)

4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H(3) Receptor Agonists with in Vivo Central Nervous System Activity

di Wágner, Gábor, Mocking, Tamara A. M., Arimont, Marta, Provensi, Gustavo, Rani, Barbara, Silva-Marques, Bruna, Latacz, Gniewomir, Da Costa Pereira, Daniel, Karatzidou, Christina, Vischer, Henry F., Wijtmans, Maikel, Kieć-Kononowicz, Katarzyna, de Esch, Iwan J. P., Leurs, Rob
Pubblicato in J Med Chem (2019)

Inhibition of autotransporter biogenesis by small molecules

di Steenhuis, Maurice, Abdallah, Abdallah M., de Munnik, Sabrina M., Kuhne, Sebastiaan, Sterk, Geert‐Jan, van den Berg van Saparoea, Bart, Westerhausen, Sibel, Wagner, Samuel, van der Wel, Nicole N., Wijtmans, Maikel, van Ulsen, Peter, Jong, Wouter S. P., Luirink, Joen
Pubblicato in Mol Microbiol (2019)

Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR Photopharmacology

di Hauwert, Niels J., Mocking, Tamara A. M., Da Costa Pereira, Daniel, Kooistra, Albert J., Wijnen, Lisa M., Vreeker, Gerda C. M., Verweij, Eléonore W. E., De Boer, Albertus H., Smit, Martine J., De Graaf, Chris, Vischer, Henry F., de Esch, Iwan J. P., Wijtmans, Maikel, Leurs, Rob
Pubblicato in J Am Chem Soc (2018)

Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity

di Blaazer, Antoni R., Singh, Abhimanyu K., de Heuvel, Erik, Edink, Ewald, Orrling, Kristina M., Veerman, Johan J. N., van den Bergh, Toine, Jansen, Chimed, Balasubramaniam, Erin, Mooij, Wouter J., Custers, Hans, Sijm, Maarten, Tagoe, Daniel N. A., Kalejaiye, Titilola D., Munday, Jane C., Tenor, Hermann, Matheeussen, An, Wijtmans, Maikel, Siderius, Marco, de Graaf, Chris, Maes, Louis, de Koning, Harry P., Bailey, David S., Sterk, Geert Jan, de Esch, Iwan J. P., Brown, David G., Leurs, Rob
Pubblicato in J Med Chem (2018)