SARS-CoV-2 Entry Inhibitors: Small Molecules and Peptides Targeting Virus or Host Cells

gan Cannalire, Rolando, Stefanelli, Irina, Cerchia, Carmen, Beccari, Andrea R., Pelliccia, Sveva, Summa, Vincenzo
Cyhoeddwyd yn Int J Mol Sci (2020)

Targeting SARS-CoV-2 Proteases and Polymerase for COVID-19 Treatment: State of the Art and Future Opportunities

gan Cannalire, Rolando, Cerchia, Carmen, Beccari, Andrea R., Di Leva, Francesco Saverio, Summa, Vincenzo
Cyhoeddwyd yn J Med Chem (2020)

Visible-Light Photocatalytic Functionalization of Isocyanides for the Synthesis of Secondary Amides and Ketene Aminals

gan Cannalire, Rolando, Amato, Jussara, Summa, Vincenzo, Novellino, Ettore, Tron, Gian Cesare, Giustiniano, Mariateresa
Cyhoeddwyd yn J Org Chem (2020)

Synthesis and Antiproliferative Activity of Nitric Oxide-Donor Largazole Prodrugs

gan Borgini, Matteo, Zamperini, Claudio, Poggialini, Federica, Ferrante, Luca, Summa, Vincenzo, Botta, Maurizio, Fabio, Romano Di
Cyhoeddwyd yn ACS Med Chem Lett (2020)

Salivary Metabolome and Soccer Match: Challenges for Understanding Exercise induced Changes

gan Pitti, Erica, Petrella, Greta, Di Marino, Sara, Summa, Vincenzo, Perrone, Marco, D’Ottavio, Stefano, Bernardini, Andrea, Cicero, Daniel Oscar
Cyhoeddwyd yn Metabolites (2019)

Early metabolic response to acute myocardial ischaemia in patients undergoing elective coronary angioplasty

gan Di Marino, Sara, Viceconte, Nicola, Lembo, Angelo, Summa, Vincenzo, Tanzilli, Gaetano, Raparelli, Valeria, Truscelli, Giovanni, Mangieri, Enrico, Gaudio, Carlo, Cicero, Daniel Oscar
Cyhoeddwyd yn Open Heart (2018)

6-Bromoindirubin-3′-oxime intercepts GSK3 signaling to promote and enhance skeletal muscle differentiation affecting miR-206 expression in mice

gan Ragozzino, Elvira, Brancaccio, Mariarita, Di Costanzo, Antonella, Scalabrì, Francesco, Andolfi, Gennaro, Wanderlingh, Luca G., Patriarca, Eduardo J., Minchiotti, Gabriella, Altamura, Sergio, Varrone, Francesca, Summa, Vincenzo
Cyhoeddwyd yn Sci Rep (2019)

Publisher Correction: 6-Bromoindirubin-3′-oxime intercepts GSK3 signaling to promote and enhance skeletal muscle differentiation affecting miR-206 expression in mice

gan Ragozzino, Elvira, Brancaccio, Mariarita, Di Costanzo, Antonella, Scalabrì, Francesco, Andolfi, Gennaro, Wanderlingh, Luca G., Patriarca, Eduardo J., Minchiotti, Gabriella, Altamura, Sergio, Summa, Vincenzo, Varrone, Francesca
Cyhoeddwyd yn Sci Rep (2020)

Personalized Metabolic Profile by Synergic Use of NMR and HRMS

gan Petrella, Greta, Montesano, Camilla, Lentini, Sara, Ciufolini, Giorgia, Vanni, Domitilla, Speziale, Roberto, Salonia, Andrea, Montorsi, Francesco, Summa, Vincenzo, Vago, Riccardo, Orsatti, Laura, Monteagudo, Edith, Cicero, Daniel Oscar
Cyhoeddwyd yn Molecules (2021)

Synthesis and Evaluation of Bifunctional Aminothiazoles as Antiretrovirals Targeting the HIV-1 Nucleocapsid Protein

gan Mori, Mattia, Dasso Lang, Maria Chiara, Saladini, Francesco, Palombi, Nastasja, Kovalenko, Lesia, De Forni, Davide, Poddesu, Barbara, Friggeri, Laura, Giannini, Alessia, Malancona, Savina, Summa, Vincenzo, Zazzi, Maurizio, Mely, Yves, Botta, Maurizio
Cyhoeddwyd yn ACS Med Chem Lett (2018)

Synthesis and Biological Evaluation of RGD–Cryptophycin Conjugates for Targeted Drug Delivery

gan Borbély, Adina, Figueras, Eduard, Martins, Ana, Esposito, Simone, Auciello, Giulio, Monteagudo, Edith, Di Marco, Annalise, Summa, Vincenzo, Cordella, Paola, Perego, Raffaella, Kemker, Isabell, Frese, Marcel, Gallinari, Paola, Steinkühler, Christian, Sewald, Norbert
Cyhoeddwyd yn Pharmaceutics (2019)

Identification of Isoform 2 Acid-Sensing Ion Channel Inhibitors as Tool Compounds for Target Validation Studies in CNS

gan Bencheva, Leda Ivanova, De Matteo, Marilenia, Ferrante, Luca, Ferrara, Marco, Prandi, Adolfo, Randazzo, Pietro, Ronzoni, Silvano, Sinisi, Roberta, Seneci, Pierfausto, Summa, Vincenzo, Gallo, Mariana, Veneziano, Maria, Cellucci, Antonella, Mazzocchi, Nausicaa, Menegon, Andrea, Di Fabio, Romano
Cyhoeddwyd yn ACS Med Chem Lett (2019)

Improved Selective Class I HDAC and Novel Selective HDAC3 Inhibitors: Beyond Hydroxamic Acids and Benzamides

gan Bresciani, Alberto, Ontoria, Jesus M., Biancofiore, Ilaria, Cellucci, Antonella, Ciammaichella, Alina, Di Marco, Annalise, Ferrigno, Federica, Francone, Alessandra, Malancona, Savina, Monteagudo, Edith, Nizi, Emanuela, Pace, Paola, Ponzi, Simona, Rossetti, Ilaria, Veneziano, Maria, Summa, Vincenzo, Harper, Steven
Cyhoeddwyd yn ACS Med Chem Lett (2018)

Prdm16-mediated H3K9 methylation controls fibro-adipogenic progenitors identity during skeletal muscle repair

gan Biferali, Beatrice, Bianconi, Valeria, Perez, Daniel Fernandez, Kronawitter, Sophie Pöhle, Marullo, Fabrizia, Maggio, Roberta, Santini, Tiziana, Polverino, Federica, Biagioni, Stefano, Summa, Vincenzo, Toniatti, Carlo, Pasini, Diego, Stricker, Sigmar, Di Fabio, Romano, Chiacchiera, Fulvio, Peruzzi, Giovanna, Mozzetta, Chiara
Cyhoeddwyd yn Sci Adv (2021)

Combined Peptide and Small-Molecule Approach toward Nonacidic THIQ Inhibitors of the KEAP1/NRF2 Interaction

gan Ontoria, Jesus M., Biancofiore, Ilaria, Fezzardi, Paola, Ferrigno, Federica, Torrente, Esther, Colarusso, Stefania, Bianchi, Elisabetta, Andreini, Matteo, Patsilinakos, Alexandros, Kempf, Georg, Augustin, Martin, Steinbacher, Stefan, Summa, Vincenzo, Pacifici, Robert, Muñoz-Sanjuan, Ignacio, Park, Larry, Bresciani, Alberto, Dominguez, Celia, Sherman, Leticia Toledo, Harper, Steven
Cyhoeddwyd yn ACS Med Chem Lett (2020)

Discovery of a Selective Series of Inhibitors of Plasmodium falciparum HDACs

gan Ontoria, Jesus M., Paonessa, Giacomo, Ponzi, Simona, Ferrigno, Federica, Nizi, Emanuela, Biancofiore, Ilaria, Malancona, Savina, Graziani, Rita, Roberts, David, Willis, Paul, Bresciani, Alberto, Gennari, Nadia, Cecchetti, Ottavia, Monteagudo, Edith, Orsale, Maria V., Veneziano, Maria, Di Marco, Annalise, Cellucci, Antonella, Laufer, Ralph, Altamura, Sergio, Summa, Vincenzo, Harper, Steven
Cyhoeddwyd yn ACS Med Chem Lett (2016)

5,6-Dihydroxypyrimidine Scaffold to Target HIV-1 Nucleocapsid Protein

gan Malancona, Savina, Mori, Mattia, Fezzardi, Paola, Santoriello, Marisabella, Basta, Andreina, Nibbio, Martina, Kovalenko, Lesia, Speziale, Roberto, Battista, Maria Rosaria, Cellucci, Antonella, Gennari, Nadia, Monteagudo, Edith, Di Marco, Annalise, Giannini, Alessia, Sharma, Rajhans, Pires, Manuel, Real, Eleonore, Zazzi, Maurizio, Dasso Lang, Maria Chiara, De Forni, Davide, Saladini, Francesco, Mely, Yves, Summa, Vincenzo, Harper, Steven, Botta, Maurizio
Cyhoeddwyd yn ACS Med Chem Lett (2020)

MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants

gan Summa, Vincenzo, Ludmerer, Steven W., McCauley, John A., Fandozzi, Christine, Burlein, Christine, Claudio, Giuliano, Coleman, Paul J., DiMuzio, Jillian M., Ferrara, Marco, Di Filippo, Marcello, Gates, Adam T., Graham, Donald J., Harper, Steven, Hazuda, Daria J., McHale, Carolyn, Monteagudo, Edith, Pucci, Vincenzo, Rowley, Michael, Rudd, Michael T., Soriano, Aileen, Stahlhut, Mark W., Vacca, Joseph P., Olsen, David B., Liverton, Nigel J., Carroll, Steven S.
Cyhoeddwyd 2012

MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants

gan Summa, Vincenzo, Ludmerer, Steven W., McCauley, John A., Fandozzi, Christine, Burlein, Christine, Claudio, Giuliano, Coleman, Paul J., DiMuzio, Jillian M., Ferrara, Marco, Filippo, Marcello Di, Gates, Adam T., Graham, Donald J., Harper, Steven, Hazuda, Daria J., Huang, Qian, McHale, Carolyn, Monteagudo, Edith, Pucci, Vincenzo, Rowley, Michael, Rudd, Michael T., Soriano, Aileen, Stahlhut, Mark W., Vacca, Joseph P., Olsen, David B., Liverton, Nigel J., Carroll, Steven S.
Cyhoeddwyd 2014

Identification of Inhibitors of SARS-CoV-2 3CL-Pro Enzymatic Activity Using a Small Molecule in Vitro Repurposing Screen

gan Kuzikov, Maria, Costanzi, Elisa, Reinshagen, Jeanette, Esposito, Francesca, Vangeel, Laura, Wolf, Markus, Ellinger, Bernhard, Claussen, Carsten, Geisslinger, Gerd, Corona, Angela, Iaconis, Daniela, Talarico, Carmine, Manelfi, Candida, Cannalire, Rolando, Rossetti, Giulia, Gossen, Jonas, Albani, Simone, Musiani, Francesco, Herzog, Katja, Ye, Yang, Giabbai, Barbara, Demitri, Nicola, Jochmans, Dirk, Jonghe, Steven De, Rymenants, Jasper, Summa, Vincenzo, Tramontano, Enzo, Beccari, Andrea R., Leyssen, Pieter, Storici, Paola, Neyts, Johan, Gribbon, Philip, Zaliani, Andrea
Cyhoeddwyd yn ACS Pharmacol Transl Sci (2021)