Bio-orthogonal Affinity Purification of Direct Kinase Substrates

بواسطة Allen, Jasmina J., Lazerwith, Scott E., Shokat, Kevan M.
منشور في 2005

Long Dissociation of Bictegravir from HIV-1 Integrase-DNA Complexes

بواسطة White, Kirsten L., Osman, Nathan, Cuadra-Foy, Ernesto, Brenner, Bluma G., Shivakumar, Devleena, Campigotto, Federico, Tsiang, Manuel, Morganelli, Philip A., Novikov, Nikolai, Lazerwith, Scott E., Jin, Haolun, Niedziela-Majka, Anita
الحاوية / القاعدة Antimicrob Agents Chemother (2021)

Benzothiophene piperazine and piperidine urea inhibitors of fatty acid amide hydrolase (FAAH)

بواسطة Johnson, Douglas S., Ahn, Kay, Kesten, Suzanne, Lazerwith, Scott E., Song, Yuntao, Morris, Mark, Fay, Lorraine, Gregory, Tracy, Stiff, Cory, Dunbar, James B., Liimatta, Marya, Beidler, David, Smith, Sarah, Nomanbhoy, Tyzoon K., Cravatt, Benjamin F.
منشور في 2009

A Small-Molecule Inhibitor of Hepatitis C Virus Infectivity

بواسطة Bush, Caroline O., Pokrovskii, Maria V., Saito, Roland, Morganelli, Philip, Canales, Eda, Clarke, Michael O., Lazerwith, Scott E., Golde, Justin, Reid, Brian G., Babaoglu, Kerim, Pagratis, Nikos, Zhong, Weidong, Delaney, William E., Paulson, Matthew S., Beran, Rudolf K. F.
منشور في 2014

Discovery of PF-04457845: A Highly Potent, Orally Bioavailable, and Selective Urea FAAH Inhibitor

بواسطة Johnson, Douglas S., Stiff, Cory, Lazerwith, Scott E., Kesten, Suzanne R., Fay, Lorraine K., Morris, Mark, Beidler, David, Liimatta, Marya B., Smith, Sarah E., Dudley, David T., Sadagopan, Nalini, Bhattachar, Shobha N., Kesten, Stephen J., Nomanbhoy, Tyzoon K., Cravatt, Benjamin F., Ahn, Kay
منشور في 2010

Antiviral Activity of Bictegravir (GS-9883), a Novel Potent HIV-1 Integrase Strand Transfer Inhibitor with an Improved Resistance Profile

بواسطة Tsiang, Manuel, Jones, Gregg S., Goldsmith, Joshua, Mulato, Andrew, Hansen, Derek, Kan, Elaine, Tsai, Luong, Bam, Rujuta A., Stepan, George, Stray, Kirsten M., Niedziela-Majka, Anita, Yant, Stephen R., Yu, Helen, Kukolj, George, Cihlar, Tomas, Lazerwith, Scott E., White, Kirsten L., Jin, Haolun
الحاوية / القاعدة Antimicrob Agents Chemother (2016)

Optimization of Pharmacokinetics through Manipulation of Physicochemical Properties in a Series of HCV Inhibitors

بواسطة Lazerwith, Scott E., Bahador, Gina, Canales, Eda, Cheng, Guofeng, Chong, Lee, Clarke, Michael O., Doerffler, Edward, Eisenberg, Eugene J., Hayes, Jaclyn, Lu, Bing, Liu, Qi, Matles, Mike, Mertzman, Michael, Mitchell, Michael L., Morganelli, Philip, Murray, Bernard P., Robinson, Margaret, Strickley, Robert G., Tessler, Megan, Tirunagari, Neeraj, Wang, Jianhong, Wang, Yujin, Zhang, Jennifer R., Zheng, Xubin, Zhong, Weidong, Watkins, William J.
منشور في 2011

Preclinical Characterization of GS-9669, a Thumb Site II Inhibitor of the Hepatitis C Virus NS5B Polymerase

بواسطة Fenaux, Martijn, Eng, Stacey, Leavitt, Stephanie A., Lee, Yu-Jen, Mabery, Eric M., Tian, Yang, Byun, Daniel, Canales, Eda, Clarke, Michael O., Doerffler, Edward, Lazerwith, Scott E., Lew, Willard, Liu, Qi, Mertzman, Michael, Morganelli, Philip, Xu, Lianhong, Ye, Hong, Zhang, Jennifer, Matles, Mike, Murray, Bernard P., Mwangi, Judy, Zhang, Jingyu, Hashash, Ahmad, Krawczyk, Steve H., Bidgood, Alison M., Appleby, Todd C., Watkins, William J.
منشور في 2013

Clinical targeting of HIV capsid protein with a long-acting small molecule

بواسطة Link, John O., Rhee, Martin S., Tse, Winston C., Zheng, Jim, Somoza, John R., Rowe, William, Begley, Rebecca, Chiu, Anna, Mulato, Andrew, Hansen, Derek, Singer, Eric, Tsai, Luong K., Bam, Rujuta A., Chou, Chien-Hung, Canales, Eda, Brizgys, Gediminas, Zhang, Jennifer R., Li, Jiayao, Graupe, Michael, Morganelli, Philip, Liu, Qi, Wu, Qiaoyin, Halcomb, Randall L., Saito, Roland D., Schroeder, Scott D., Lazerwith, Scott E., Bondy, Steven, Jin, Debi, Hung, Magdeleine, Novikov, Nikolai, Liu, Xiaohong, Villaseñor, Armando G., Cannizzaro, Carina E., Hu, Eric Y., Anderson, Robert L., Appleby, Todd C., Lu, Bing, Mwangi, Judy, Liclican, Albert, Niedziela-Majka, Anita, Papalia, Giuseppe A., Wong, Melanie H., Leavitt, Stephanie A., Xu, Yili, Koditek, David, Stepan, George J., Yu, Helen, Pagratis, Nikos, Clancy, Sheila, Ahmadyar, Shekeba, Cai, Terrence Z., Sellers, Scott, Wolckenhauer, Scott A., Ling, John, Callebaut, Christian, Margot, Nicolas, Ram, Renee R., Liu, Ya-Pei, Hyland, Rob, Sinclair, Gary I., Ruane, Peter J., Crofoot, Gordon E., McDonald, Cheryl K., Brainard, Diana M., Lad, Latesh, Swaminathan, Swami, Sundquist, Wesley I., Sakowicz, Roman, Chester, Anne E., Lee, William E., Daar, Eric S., Yant, Stephen R., Cihlar, Tomas
الحاوية / القاعدة Nature (2020)