Sandmeyer reaction repurposed for the site-selective, non-oxidizing radioiodination of fully-deprotected peptides: Studies on the endogenous opioid peptide α-neoendorphin

Yazar: Pickett, Julie E., Nagakura, Kunihiko, Pasternak, Anna R., Grinnell, Steven G., Majumdar, Susruta, Lewis, Jason S., Pasternak, Gavril W.
Baskı/Yayın Bilgisi 2013

Pharmacologic Characterization in the Rat of a Potent Analgesic Lacking Respiratory Depression, IBNtxA

Yazar: Grinnell, Steven G., Majumdar, Susruta, Narayan, Ankita, Le Rouzic, Valerie, Ansonoff, Michael, Pintar, John E., Pasternak, Gavril W.
Baskı/Yayın Bilgisi 2014

Synthesis and Characterization of Azido Aryl Analogs of IBNtxA for Radio-Photoaffinity Labeling Opioid Receptors in Cell Lines and in Mouse Brain

Yazar: Grinnell, Steven G., Uprety, Rajendra, Varadi, Andras, Subrath, Joan, Hunkele, Amanda, Pan, Ying Xian, Pasternak, Gavril W., Majumdar, Susruta
Yayımlandı Cell Mol Neurobiol (2020)

Novel 6β-acylaminomorphinans with analgesic activity

Yazar: Váradi, András, Hosztafi, Sándor, Rouzic, Valerie Le, Tóth, Gergő, Urai, Ákos, Noszál, Béla, Pasternak, Gavril W., Grinnell, Steven G., Majumdar, Susruta
Baskı/Yayın Bilgisi 2013

Mild, Pd-catalyzed stannylation of radioiodination targets

Yazar: Pickett, Julie E., Váradi, András, Palmer, Travis C., Grinnell, Steven G., Schrock, Joel M., Pasternak, Gavril W., Karimov, Rashad R., Majumdar, Susruta
Yayımlandı Bioorg Med Chem Lett (2015)

Truncated mu opioid GPCR variant involvement in opioid-dependent and opioid-independent pain modulatory systems within the CNS

Yazar: Marrone, Gina F., Grinnell, Steven G., Lu, Zhigang, Rossi, Grace C., Le Rouzic, Valerie, Xu, Jin, Majumdar, Susruta, Pan, Ying-Xian, Pasternak, Gavril W.
Yayımlandı Proc Natl Acad Sci U S A (2016)

Regional heterogeneity of D2-receptor signaling in the dorsal striatum and nucleus accumbens

Yazar: Marcott, Pamela F, Gong, Sheng, Donthamsetti, Prashant, Grinnell, Steven G., Nelson, Melissa N., Newman, Amy H, Birnbaumer, Lutz, Martemyanov, Kirill A, Javitch, Jonathan A, Ford, Christopher P
Yayımlandı Neuron (2018)

Mediation of buprenorphine analgesia by a combination of traditional and truncated mu opioid receptor splice variants

Yazar: Grinnell, Steven G., Ansonoff, Michael, Marrone, Gina F., Lu, Zhigang, Narayan, Ankita, Xu, Jin, Rossi, Grace, Majumdar, Susruta, Pan, Ying-Xian, Bassoni, Daniel L., Pintar, John, Pasternak, Gavril
Yayımlandı Synapse (2016)

7-Hydroxymitragynine Is an Active Metabolite of Mitragynine and a Key Mediator of Its Analgesic Effects

Yazar: Kruegel, Andrew C., Uprety, Rajendra, Grinnell, Steven G., Langreck, Cory, Pekarskaya, Elizabeth A., Le Rouzic, Valerie, Ansonoff, Michael, Gassaway, Madalee M., Pintar, John E., Pasternak, Gavril W., Javitch, Jonathan A., Majumdar, Susruta, Sames, Dalibor
Yayımlandı ACS Cent Sci (2019)

The Behavioral Effects of the Antidepressant Tianeptine Require the Mu-Opioid Receptor

Yazar: Samuels, Benjamin Adam, Nautiyal, Katherine M, Kruegel, Andrew C, Levinstein, Marjorie R, Magalong, Valerie M, Gassaway, Madalee M, Grinnell, Steven G, Han, Jaena, Ansonoff, Michael A, Pintar, John E, Javitch, Jonathan A, Sames, Dalibor, Hen, René
Yayımlandı Neuropsychopharmacology (2017)

Mitragynine/Corynantheidine Pseudoindoxyls As Opioid Analgesics with Mu Agonism and Delta Antagonism, Which Do Not Recruit β-Arrestin-2

Yazar: Váradi, András, Marrone, Gina F., Palmer, Travis C., Narayan, Ankita, Szabó, Márton R., Le Rouzic, Valerie, Grinnell, Steven G., Subrath, Joan J., Warner, Evelyn, Kalra, Sanjay, Hunkele, Amanda, Pagirsky, Jeremy, Eans, Shainnel O., Medina, Jessica M., Xu, Jin, Pan, Ying-Xian, Borics, Attila, Pasternak, Gavril W., McLaughlin, Jay P., Majumdar, Susruta
Yayımlandı J Med Chem (2016)

Controlling opioid receptor functional selectivity by targeting distinct subpockets of the orthosteric site

Yazar: Uprety, Rajendra, Che, Tao, Zaidi, Saheem A, Grinnell, Steven G, Varga, Balázs R, Faouzi, Abdelfattah, Slocum, Samuel T, Allaoa, Abdullah, Varadi, András, Nelson, Melissa, Bernhard, Sarah M, Kulko, Elizaveta, Le Rouzic, Valerie, Eans, Shainnel O, Simons, Chloe A, Hunkele, Amanda, Subrath, Joan, Pan, Ying Xian, Javitch, Jonathan A, McLaughlin, Jay P, Roth, Bryan L, Pasternak, Gavril W, Katritch, Vsevolod, Majumdar, Susruta
Yayımlandı eLife (2021)