Synthesis of spiro-2,6-dioxopiperazine and spiro-2,6-dioxopyrazine scaffolds using amino acids in a three-component reaction to generate potential Sigma-1 (σ1) receptor selective l...

od Uprety, Rajendra, Varadi, Andras, Allaoa, Abdullah, Redel-Traub, Gabriel N., Palmer, Travis C., Feinberg, Evan N., Ferris, Alex C., Pande, Vijay S., Pasternak, Gavril W., Majumdar, Susruta
izdano v Eur J Med Chem (2018)

Synthesis and Pharmacology of a Novel μ–δ Opioid Receptor Heteromer-Selective Agonist Based on the Carfentanyl Template

od Faouzi, Abdelfattah, Uprety, Rajendra, Gomes, Ivone, Massaly, Nicolas, Keresztes, Attila I., Le Rouzic, Valerie, Gupta, Achla, Zhang, Tiffany, Yoon, Hye Jean, Ansonoff, Michael, Allaoa, Abdullah, Pan, Ying Xian, Pintar, John, Morón, Jose A., Streicher, John M., Devi, Lakshmi A., Majumdar, Susruta
izdano v J Med Chem (2020)

Controlling opioid receptor functional selectivity by targeting distinct subpockets of the orthosteric site

od Uprety, Rajendra, Che, Tao, Zaidi, Saheem A, Grinnell, Steven G, Varga, Balázs R, Faouzi, Abdelfattah, Slocum, Samuel T, Allaoa, Abdullah, Varadi, András, Nelson, Melissa, Bernhard, Sarah M, Kulko, Elizaveta, Le Rouzic, Valerie, Eans, Shainnel O, Simons, Chloe A, Hunkele, Amanda, Subrath, Joan, Pan, Ying Xian, Javitch, Jonathan A, McLaughlin, Jay P, Roth, Bryan L, Pasternak, Gavril W, Katritch, Vsevolod, Majumdar, Susruta
izdano v eLife (2021)