Extent of Helical Induction Caused by Introducing α-Aminoisobutyric Acid into an Oligovaline Sequence

по Tsuji, Genichiro, Misawa, Takashi, Doi, Mitsunobu, Demizu, Yosuke
Опубликовано в: ACS Omega (2018)

Selective Degradation of Target Proteins by Chimeric Small-Molecular Drugs, PROTACs and SNIPERs

по Ishikawa, Minoru, Tomoshige, Shusuke, Demizu, Yosuke, Naito, Mikihiko
Опубликовано в: Pharmaceuticals (Basel) (2020)

NAD-dependent isocitrate dehydrogenase as a novel target of tributyltin in human embryonic carcinoma cells

по Yamada, Shigeru, Kotake, Yaichiro, Demizu, Yosuke, Kurihara, Masaaki, Sekino, Yuko, Kanda, Yasunari
Опубликовано 2014

A synthetic cannabinoid FDU-NNEI, two 2H-indazole isomers of synthetic cannabinoids AB-CHMINACA and NNEI indazole analog (MN-18), a phenethylamine derivative N–OH-EDMA, and a cathi...

по Uchiyama, Nahoko, Shimokawa, Yoshihiko, Kikura-Hanajiri, Ruri, Demizu, Yosuke, Goda, Yukihiro, Hakamatsuka, Takashi
Опубликовано в: Forensic Toxicol (2015)

Rational design of novel amphipathic antimicrobial peptides focused on the distribution of cationic amino acid residues

по Misawa, Takashi, Goto, Chihiro, Shibata, Norihito, Hirano, Motoharu, Kikuchi, Yutaka, Naito, Mikihiko, Demizu, Yosuke
Опубликовано в: Medchemcomm (2019)

Development of Antimicrobial Stapled Peptides Based on Magainin 2 Sequence

по Hirano, Motoharu, Saito, Chihiro, Yokoo, Hidetomo, Goto, Chihiro, Kawano, Ryuji, Misawa, Takashi, Demizu, Yosuke
Опубликовано в: Molecules (2021)

Targeted Protein Degradation by Chimeric Compounds using Hydrophobic E3 Ligands and Adamantane Moiety

по Shoda, Takuji, Ohoka, Nobumichi, Tsuji, Genichiro, Fujisato, Takuma, Inoue, Hideshi, Demizu, Yosuke, Naito, Mikihiko, Kurihara, Masaaki
Опубликовано в: Pharmaceuticals (Basel) (2020)

Design, Synthesis, and Biological Activity of Conformationally Restricted Analogues of Silibinin

по Mizuno, Mirei, Mori, Kazunori, Tsuchiya, Keisuke, Takaki, Takashi, Misawa, Takashi, Demizu, Yosuke, Shibanuma, Motoko, Fukuhara, Kiyoshi
Опубликовано в: ACS Omega (2020)

Development of a Hematopoietic Prostaglandin D Synthase-Degradation Inducer

по Yokoo, Hidetomo, Shibata, Norihito, Naganuma, Miyako, Murakami, Yuki, Fujii, Kiyonaga, Ito, Takahito, Aritake, Kosuke, Naito, Mikihiko, Demizu, Yosuke
Опубликовано в: ACS Med Chem Lett (2021)

Development of ciclesonide analogues that block SARS-CoV-2 RNA replication

по Tsuji, Genichiro, Yonemitsu, Kenzo, Ito, Takahito, Yanase, Yuta, Uema, Masashi, Ohoka, Nobumichi, Inoue, Takao, Asakura, Hiroshi, Demizu, Yosuke
Опубликовано в: Bioorg Med Chem Lett (2021)

Development of hybrid small molecules that induce degradation of estrogen receptor‐alpha and necrotic cell death in breast cancer cells

по Okuhira, Keiichiro, Demizu, Yosuke, Hattori, Takayuki, Ohoka, Nobumichi, Shibata, Norihito, Nishimaki‐Mogami, Tomoko, Okuda, Haruhiro, Kurihara, Masaaki, Naito, Mikihiko
Опубликовано в: Cancer Sci (2013)

Development of a Cell-penetrating Peptide that Exhibits Responsive Changes in its Secondary Structure in the Cellular Environment

по Yamashita, Hiroko, Kato, Takuma, Oba, Makoto, Misawa, Takashi, Hattori, Takayuki, Ohoka, Nobumichi, Tanaka, Masakazu, Naito, Mikihiko, Kurihara, Masaaki, Demizu, Yosuke
Опубликовано в: Sci Rep (2016)

Design, synthesis, and anti-HIV-1 activity of 1-aromatic methyl-substituted 3-(3,5-dimethylbenzyl)uracil and N-3,5-dimethylbenzyl-substituted urea derivatives

по Sakakibara, Norikazu, Baba, Masanori, Okamoto, Mika, Toyama, Masaaki, Demizu, Yosuke, Misawa, Takashi, Kurihara, Masaaki, Irie, Kohji, Kato, Yoshihisa, Maruyama, Tokumi
Опубликовано в: Antivir Chem Chemother (2015)

Development of Agonist-Based PROTACs Targeting Liver X Receptor

по Xu, Hanqiao, Ohoka, Nobumichi, Yokoo, Hidetomo, Nemoto, Kanako, Ohtsuki, Takashi, Matsufuji, Hiroshi, Naito, Mikihiko, Inoue, Takao, Tsuji, Genichiro, Demizu, Yosuke
Опубликовано в: Front Chem (2021)

Design and synthesis of novel selective estrogen receptor degradation inducers based on the diphenylheptane skeleton

по Misawa, Takashi, Fujisato, Takuma, Kanda, Yasunari, Ohoka, Nobumichi, Shoda, Takuji, Yorioka, Momoko, Makishima, Makoto, Sekino, Yuko, Naito, Mikihiko, Demizu, Yosuke, Kurihara, Masaaki
Опубликовано в: Medchemcomm (2016)

Critical role of mitochondrial ubiquitination and the OPTN–ATG9A axis in mitophagy

по Yamano, Koji, Kikuchi, Reika, Kojima, Waka, Hayashida, Ryota, Koyano, Fumika, Kawawaki, Junko, Shoda, Takuji, Demizu, Yosuke, Naito, Mikihiko, Tanaka, Keiji, Matsuda, Noriyuki
Опубликовано в: J Cell Biol (2020)

Design, synthesis, and anti-HIV-1 activity of 1-substituted 3-(3,5-dimethylbenzyl)triazine derivatives

по Sakakibara, Norikazu, Balboni, Gianfranco, Congiu, Cenzo, Onnis, Valentina, Demizu, Yosuke, Misawa, Takashi, Kurihara, Masaaki, Kato, Yoshihisa, Maruyama, Tokumi, Toyama, Masaaki, Okamoto, Mika, Baba, Masanori
Опубликовано в: Antivir Chem Chemother (2015)

Rapid and efficient high-performance liquid chromatography analysis of N-nitrosodimethylamine impurity in valsartan drug substance and its products

по Masada, Sayaka, Tsuji, Genichiro, Arai, Ryoko, Uchiyama, Nahoko, Demizu, Yosuke, Tsutsumi, Tomoaki, Abe, Yasuhiro, Akiyama, Hiroshi, Hakamatsuka, Takashi, Izutsu, Ken-ichi, Goda, Yukihiro, Okuda, Haruhiro
Опубликовано в: Sci Rep (2019)

Identification of embryonic precursor cells that differentiate into thymic epithelial cells expressing autoimmune regulator

по Akiyama, Nobuko, Takizawa, Nobukazu, Miyauchi, Maki, Yanai, Hiromi, Tateishi, Ryosuke, Shinzawa, Miho, Yoshinaga, Riko, Kurihara, Masaaki, Demizu, Yosuke, Yasuda, Hisataka, Yagi, Shintaro, Wu, Guoying, Matsumoto, Mitsuru, Sakamoto, Reiko, Yoshida, Nobuaki, Penninger, Josef M., Kobayashi, Yasuhiro, Inoue, Jun-ichiro, Akiyama, Taishin
Опубликовано в: J Exp Med (2016)