A balance between elongation and trimming regulates telomere stability in stem cells

по Rivera, Teresa, Haggblom, Candy, Cosconati, Sandro, Karlseder, Jan
Опубликовано в: Nat Struct Mol Biol (2016)

Structure-Based Virtual Screening and Biological Evaluation of Mycobacterium tuberculosis Adenosine 5′-Phosphosulfate Reductase Inhibitors

по Cosconati, Sandro, Hong, Jiyoung A., Novellino, Ettore, Carroll, Kate S, Goodsell, David S., Olson, Arthur J
Опубликовано 2008

Virtual Screening with AutoDock: Theory and Practice

по Cosconati, Sandro, Forli, Stefano, Perryman, Alex L., Harris, Rodney, Goodsell, David S., Olson, Arthur J.
Опубликовано 2010

Olive Leaves and Hibiscus Flowers Extracts-Based Preparation Protect Brain from Oxidative Stress-Induced Injury

по Chiaino, Elda, Micucci, Matteo, Cosconati, Sandro, Novellino, Ettore, Budriesi, Roberta, Chiarini, Alberto, Frosini, Maria
Опубликовано в: Antioxidants (Basel) (2020)

Synthesis and Gene Silencing Properties of siRNAs Containing Terminal Amide Linkages

по Gaglione, Maria, Mercurio, M. Emilia, Potenza, Nicoletta, Mosca, Nicola, Russo, Aniello, Novellino, Ettore, Cosconati, Sandro, Messere, Anna
Опубликовано 2014

Endogenous vs Exogenous Allosteric Modulators in GPCRs: A dispute for shuttling CB(1) among different membrane microenvironments

по Stornaiuolo, Mariano, Bruno, Agostino, Botta, Lorenzo, Regina, Giuseppe La, Cosconati, Sandro, Silvestri, Romano, Marinelli, Luciana, Novellino, Ettore
Опубликовано в: Sci Rep (2015)

Identification of novel indole derivatives acting as inhibitors of the Keap1–Nrf2 interaction

по Cosimelli, Barbara, Greco, Giovanni, Laneri, Sonia, Novellino, Ettore, Sacchi, Antonia, Amendola, Giorgio, Cosconati, Sandro, Bortolozzi, Roberta, Viola, Giampietro
Опубликовано в: J Enzyme Inhib Med Chem (2019)

Tuning RNA Interference by Enhancing siRNA/PAZ Recognition

по Gaglione, Maria, Potenza, Nicoletta, Di Fabio, Giovanni, Romanucci, Valeria, Mosca, Nicola, Russo, Aniello, Novellino, Ettore, Cosconati, Sandro, Messere, Anna
Опубликовано 2012

Sampling protein motion and solvent effect during ligand binding

по Limongelli, Vittorio, Marinelli, Luciana, Cosconati, Sandro, La Motta, Concettina, Sartini, Stefania, Mugnaini, Laura, Da Settimo, Federico, Novellino, Ettore, Parrinello, Michele
Опубликовано 2012

3-(Fur-2-yl)-10-(2-phenylethyl)-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one, a Novel Adenosine Receptor Antagonist with A(2A)-Mediated Neuroprotective Effects

по Scatena, Alessia, Fornai, Francesco, Trincavelli, Maria Letizia, Taliani, Sabrina, Daniele, Simona, Pugliesi, Isabella, Cosconati, Sandro, Martini, Claudia, Da Settimo, Federico
Опубликовано 2011

Protein Flexibility in Virtual Screening: The BACE-1 Case Study

по Cosconati, Sandro, Marinelli, Luciana, Di Leva, Francesco Saverio, La Pietra, Valeria, De Simone, Angela, Mancini, Francesca, Andrisano, Vincenza, Novellino, Ettore, Goodsell, David S., Olson, Arthur J.
Опубликовано 2012

Studies on enantioselectivity of chiral 4-acetylamino-6-alkyloxy-2-alkylthiopyrimidines acting as antagonists of the human A(3) adenosine receptor

по Cosimelli, Barbara, Greco, Giovanni, Laneri, Sonia, Novellino, Ettore, Sacchi, Antonia, Collina, Simona, Rossi, Daniela, Cosconati, Sandro, Barresi, Elisabetta, Taliani, Sabrina, Trincavelli, Maria Letizia, Martini, Claudia
Опубликовано в: Medchemcomm (2017)

Two novel SIRT1 activators, SCIC2 and SCIC2.1, enhance SIRT1-mediated effects in stress response and senescence

по Scisciola, Lucia, Sarno, Federica, Carafa, Vincenzo, Cosconati, Sandro, Di Maro, Salvatore, Ciuffreda, Loreta, De Angelis, Antonella, Stiuso, Paola, Feoli, Alessandra, Sbardella, Gianluca, Altucci, Lucia, Nebbioso, Angela
Опубликовано в: Epigenetics (2020)

Decoration of chondroitin polysaccharide with threonine: synthesis, conformational study and ice-recrystallization inhibition activity

по Laezza, Antonio, Casillo, Angela, Cosconati, Sandro, Biggs, Caroline I., Fabozzi, Antonio, Paduano, Luigi, Iadonisi, Alfonso, Novellino, Ettore, Gibson, Matthew I., Randazzo, Antonio, Corsaro, Maria M., Bedini, Emiliano
Опубликовано в: Biomacromolecules (2017)

Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies

по Milite, Ciro, Amendola, Giorgio, Nocentini, Alessio, Bua, Silvia, Cipriano, Alessandra, Barresi, Elisabetta, Feoli, Alessandra, Novellino, Ettore, Da Settimo, Federico, Supuran, Claudiu T., Castellano, Sabrina, Cosconati, Sandro, Taliani, Sabrina
Опубликовано в: J Enzyme Inhib Med Chem (2019)

Discovery of Pyrido[3′,2′:5,6]thiopyrano[4,3-d]pyrimidine-Based Antiproliferative Multikinase Inhibitors

по Salerno, Silvia, Barresi, Elisabetta, García-Argáez, Aída Nelly, Taliani, Sabrina, Simorini, Francesca, Amendola, Giorgio, Tomassi, Stefano, Cosconati, Sandro, Novellino, Ettore, Da Settimo, Federico, Marini, Anna Maria, Dalla Via, Lisa
Опубликовано в: ACS Med Chem Lett (2019)

Discovery of a Novel Chemotype of Histone Lysine Methyltransferase EHMT1/2 (GLP/G9a) Inhibitors: Rational Design, Synthesis, Biological Evaluation, and Co-crystal Structure

по Milite, Ciro, Feoli, Alessandra, Horton, John R., Rescigno, Donatella, Cipriano, Alessandra, Pisapia, Vincenzo, Viviano, Monica, Pepe, Giacomo, Amendola, Giorgio, Novellino, Ettore, Cosconati, Sandro, Cheng, Xiaodong, Castellano, Sabrina, Sbardella, Gianluca
Опубликовано в: J Med Chem (2019)

Structure-activity relationship of the exopolysaccharide from a psychrophilic bacterium: a strategy for cryoprotection

по Casillo, Angela, Parrilli, Ermenegilda, Sannino, Filomena, Mitchell, Daniel E., Gibson, Matthew I., Marino, Gennaro, Lanzetta, Rosa, Parrilli, Michelangelo, Cosconati, Sandro, Novellino, Ettore, Randazzo, Antonio, Tutino, Maria L., Corsaro, M. Michela
Опубликовано в: Carbohydr Polym (2016)

Identification of Highly Conserved Residues Involved in Inhibition of HIV-1 RNase H Function by Diketo Acid Derivatives

по Corona, Angela, Di Leva, Francesco Saverio, Thierry, Sylvain, Pescatori, Luca, Cuzzucoli Crucitti, Giuliana, Subra, Frederic, Delelis, Olivier, Esposito, Francesca, Rigogliuso, Giuseppe, Costi, Roberta, Cosconati, Sandro, Novellino, Ettore, Di Santo, Roberto, Tramontano, Enzo
Опубликовано 2014

Antitumor efficacy of Kisspeptin in human malignant mesothelioma cells

по Ciaramella, Vincenza, Della Corte, Carminia Maria, Di Mauro, Concetta, Tomassi, Stefano, Di Maro, Salvatore, Troiani, Teresa, Martinelli, Erika, Bianco, Roberto, Cosconati, Sandro, Pierantoni, Riccardo, Meccariello, Rosaria, Chianese, Rosanna, Ciardiello, Fortunato, Morgillo, Floriana
Опубликовано в: Oncotarget (2018)