Beyond radio-displacement techniques for Identification of CB(1) Ligands: The First Application of a Fluorescence-quenching Assay

by Bruno, Agostino, Lembo, Francesca, Novellino, Ettore, Stornaiuolo, Mariano, Marinelli, Luciana
Published 2014

Membrane-Sensitive Conformational States of Helix 8 in the Metabotropic Glu2 Receptor, a Class C GPCR

by Bruno, Agostino, Costantino, Gabriele, de Fabritiis, Gianni, Pastor, Manuel, Selent, Jana
Published 2012

Correction: Membrane-Sensitive Conformational States of Helix 8 in the Metabotropic Glu2 Receptor, a Class C GPCR

by Bruno, Agostino, Costantino, Gabriele, de Fabritiis, Gianni, Pastor, Manuel, Selent, Jana
Published 2012

The Glycan Role in the Glycopeptide Immunogenicity Revealed by Atomistic Simulations and Spectroscopic Experiments on the Multiple Sclerosis Biomarker CSF114(Glc)

by Bruno, Agostino, Scrima, Mario, Novellino, Ettore, D'Errico, Gerardino, D'Ursi, Anna Maria, Limongelli, Vittorio
Published in Sci Rep (2015)

Endogenous vs Exogenous Allosteric Modulators in GPCRs: A dispute for shuttling CB(1) among different membrane microenvironments

by Stornaiuolo, Mariano, Bruno, Agostino, Botta, Lorenzo, Regina, Giuseppe La, Cosconati, Sandro, Silvestri, Romano, Marinelli, Luciana, Novellino, Ettore
Published in Sci Rep (2015)

Biochemical Characterization of Aspergillus fumigatus AroH, a Putative Aromatic Amino Acid Aminotransferase

by Dindo, Mirco, Costanzi, Egidia, Pieroni, Marco, Costantini, Claudio, Annunziato, Giannamaria, Bruno, Agostino, Keller, Nancy P., Romani, Luigina, Zelante, Teresa, Cellini, Barbara
Published in Front Mol Biosci (2018)

Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor

by Magalhães, Joana, Franko, Nina, Raboni, Samanta, Annunziato, Giannamaria, Tammela, Päivi, Bruno, Agostino, Bettati, Stefano, Mozzarelli, Andrea, Pieroni, Marco, Campanini, Barbara, Costantino, Gabriele
Published in ACS Med Chem Lett (2020)

Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design

by Magalhães, Joana, Franko, Nina, Annunziato, Giannamaria, Welch, Martin, Dolan, Stephen K., Bruno, Agostino, Mozzarelli, Andrea, Armao, Stefano, Jirgensons, Aigars, Pieroni, Marco, Costantino, Gabriele, Campanini, Barbara
Published in J Enzyme Inhib Med Chem (2018)

Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases

by Annunziato, Giannamaria, Giovati, Laura, Angeli, Andrea, Pavone, Marialaura, Del Prete, Sonia, Pieroni, Marco, Capasso, Clemente, Bruno, Agostino, Conti, Stefania, Magliani, Walter, Supuran, Claudiu T., Costantino, Gabriele
Published in J Enzyme Inhib Med Chem (2018)

Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvan...

by Magalhães, Joana, Franko, Nina, Raboni, Samanta, Annunziato, Giannamaria, Tammela, Päivi, Bruno, Agostino, Bettati, Stefano, Armao, Stefano, Spadini, Costanza, Cabassi, Clotilde Silvia, Mozzarelli, Andrea, Pieroni, Marco, Campanini, Barbara, Costantino, Gabriele
Published in Pharmaceuticals (Basel) (2021)

The Aryl Hydrocarbon Receptor (AhR) Mediates the Counter-Regulatory Effects of Pelargonidins in Models of Inflammation and Metabolic Dysfunctions

by Biagioli, Michele, Carino, Adriana, Fiorucci, Chiara, Annunziato, Giannamaria, Marchianò, Silvia, Bordoni, Martina, Roselli, Rosalinda, Giorgio, Cristina Di, Castiglione, Federica, Ricci, Patrizia, Bruno, Agostino, Faccini, Andrea, Distrutti, Eleonora, Baldoni, Monia, Costantino, Gabriele, Fiorucci, Stefano
Published in Nutrients (2019)

Molecular mechanism and functional role of brefeldin A-mediated ADP-ribosylation of CtBP1/BARS

by Colanzi, Antonino, Grimaldi, Giovanna, Catara, Giuliana, Valente, Carmen, Cericola, Claudia, Liberali, Prisca, Ronci, Maurizio, Lalioti, Vasiliki S., Bruno, Agostino, Beccari, Andrea R., Urbani, Andrea, De Flora, Antonio, Nardini, Marco, Bolognesi, Martino, Luini, Alberto, Corda, Daniela
Published 2013

Binding of the Anti-FIV Peptide C8 to Differently Charged Membrane Models: From First Docking to Membrane Tubulation

by Di Marino, Daniele, Bruno, Agostino, Grimaldi, Manuela, Scrima, Mario, Stillitano, Ilaria, Amodio, Giuseppina, Della Sala, Grazia, Romagnoli, Alice, De Santis, Augusta, Moltedo, Ornella, Remondelli, Paolo, Boccia, Giovanni, D'Errico, Gerardino, D'Ursi, Anna Maria, Limongelli, Vittorio
Published in Front Chem (2020)

Everolimus induces Met inactivation by disrupting the FKBP12/Met complex

by Raimondo, Lucia, D'Amato, Valentina, Servetto, Alberto, Rosa, Roberta, Marciano, Roberta, Formisano, Luigi, Mauro, Concetta Di, Orsini, Roberta Clara, Cascetta, Priscilla, Ciciola, Paola, De Maio, Ana Paula, Di Renzo, Maria Flavia, Cosconati, Sandro, Bruno, Agostino, Randazzo, Antonio, Napolitano, Filomena, Montuori, Nunzia, Veneziani, Bianca Maria, Placido, Sabino De, Bianco, Roberto
Published in Oncotarget (2016)

Targeting the minor pocket of C5aR for the rational design of an oral allosteric inhibitor for inflammatory and neuropathic pain relief

by Moriconi, Alessio, Cunha, Thiago M., Souza, Guilherme R., Lopes, Alexandre H., Cunha, Fernando Q., Carneiro, Victor L., Pinto, Larissa G., Brandolini, Laura, Aramini, Andrea, Bizzarri, Cinzia, Bianchini, Gianluca, Beccari, Andrea R., Fanton, Marco, Bruno, Agostino, Costantino, Gabriele, Bertini, Riccardo, Galliera, Emanuela, Locati, Massimo, Ferreira, Sérgio H., Teixeira, Mauro M., Allegretti, Marcello
Published in Proc Natl Acad Sci U S A (2014)