Synthesis, Optimization and Structure-Activity Relationships of 3,5-Disubstituted Isoxazolines as New Anti-tuberculosis Agents

Por Rakesh, Dianqing Sun, Lee, Robin B., Tangallapally, Rajendra, Lee, Richard E.
Publicado em 2008

Development of CXCR4 modulators based on the lead compound RB-108

Por Bai, Renren, Jie, Xiaokang, Sun, Jian, Liang, Zhongxing, Yoon, Younghyoun, Feng, Amber, Oum, Yoonhyeun, Yu, Wenyan, Wu, Rui, Sun, Bin, Salgado, Eric, Xie, Yuanyuan, Shim, Hyunsuk
Publicado no Eur J Med Chem (2019)

New Insights into Structure–Activity Relationship of Ipomoeassin F from Its Bioisosteric 5-Oxa/Aza Analogues

Por Zong, Guanghui, Sun, Xianwei, Bhakta, Rima, Whisenhunt, Lucas, Hu, Zhijian, Wang, Feng, Shi, Wei Q.
Publicado no Eur J Med Chem (2017)

Preparation and evaluation of tetrabenazine enantiomers and all eight stereoisomers of dihydrotetrabenazine as VMAT2 inhibitors

Por Yao, Zhangyu, Wei, Xueying, Wu, Xiaoming, Katz, Jonathan L., Kopajtic, Theresa, Greig, Nigel H., Sun, Hongbin
Publicado no Eur J Med Chem (2011)

Synthesis, evaluation, and CoMFA study of fluoroquinophenoxazine derivatives as bacterial topoisomerase IA inhibitors

Por Yu, Xufen, Zhang, Mingming, Annamalai, Arasu, Bansod, Priyanka, Narula, Gagandeep, Tse-Dinh, Yuk-Ching, Sun, Dianqing
Publicado no Eur J Med Chem (2016)

Monocarbonyl analogs of curcumin inhibit growth of antibiotic sensitive and resistant strains of Mycobacterium tuberculosis

Por Baldwin, Patrick R., Reeves, Analise Z., Powell, Kimberly R., Napier, Ruth J., Swimm, Alyson I., Sun, Aiming, Giesler, Kyle, Bommarius, Bettina, Shinnick, Thomas M., Snyder, James P., Liotta, Dennis C., Kalman, Daniel
Publicado no Eur J Med Chem (2015)

Anti-inflammatory hybrids of secondary amines and amide-sulfamide derivatives

Por Bai, Renren, Sun, Jian, Liang, Zhongxing, Yoon, Younghyoun, Salgado, Eric, Feng, Amber, Oum, Yoonhyeun, Xie, Yuanyuan, Shim, Hyunsuk
Publicado no Eur J Med Chem (2018)

Synthesis and structure-activity relationship studies of novel 3,9-substituted α-carboline derivatives with high cytotoxic activity against colorectal cancer cells

Por Lin, Yi-Chien, Chen, Yi-Fong, Tseng, Li-Shin, Lee, Yueh-Hsuan, Morris-Natschke, Susan L, Kuo, Sheng-Chu, Yang, Ning-Sun, Lee, Kuo-Hsiung, Huang, Li-Jiau
Publicado no Eur J Med Chem (2016)

Hydrogen Peroxide Activated Quinone Methide Precursors with Enhanced DNA Cross-Linking Capability and Cytotoxicity towards Cancer Cells

Por Wang, Yibin, Fan, Heli, Balakrishnan, Kumudha, Lin, Zechao, Cao, Sheng, Chen, Wenbing, Fan, Yukai, Guthrie, Quibria A., Sun, Huabing, Teske, Kelly A., Gandhi, Varsha, Arnold, Leggy A., Peng, Xiaohua
Publicado no Eur J Med Chem (2017)

Synthesis and biological evaluations of chalcones, flavones and chromenes as farnesoid x receptor (FXR) antagonists

Por Zhang, Guoning, Liu, Shuainan, Tan, Wenjuan, Verma, Ruchi, Chen, Yuan, Sun, Deyang, Huan, Yi, Jiang, Qian, Wang, Xing, Wang, Na, Xu, Yang, Wong, Chiwai, Shen, Zhufang, Deng, Ruitang, Liu, Jinsong, Zhang, Yanqiao, Fang, Weishuo
Publicado no Eur J Med Chem (2017)