Understanding the structural requirements of 4-anilidopiperidine analogues for biological activities at μ and δ opioid receptors

Por Lee, Yeon Sun, Nyberg, Joel, Moye, Sharif, Agnes, Richard S., Davis, Peg, Ma, Shou-wu, Lai, Josephine, Porreca, Frank, Vardanyan, Ruben, Hruby, Victor J.
Publicado em 2007

Structure-activity relationships of non-opioid [des-Arg(7)]-dynorphin A analogues for bradykinin receptors

Por Lee, Yeon Sun, Rankin, David, Hall, Sara M., Ramos-Colon, Cyf, Ortiz, Jose Juan, Kupp, Robert, Porreca, Frank, Lai, Josephine, Hruby, Victor J.
Publicado no Bioorg Med Chem Lett (2014)

A Potent Small-Molecule Inhibitor of the MDM2-p53 Interaction (MI-888) Achieved Complete and Durable Tumor Regression in Mice

Por Zhao, Yujun, Yu, Shanghai, Sun, Wei, Liu, Liu, Lu, Jianfeng, McEachern, Donna, Shargary, Sanjeev, Bernard, Denzil, Li, Xiaoqin, Zhao, Ting, Zou, Peng, Sun, Duxin, Wang, Shaomeng
Publicado em 2013

Potent Bivalent Smac Mimetics: Effect of the Linker on Binding to Inhibitor of Apoptosis Proteins (IAPs) and Anticancer Activity

Por Sun, Haiying, Liu, Liu, Lu, Jianfeng, Bai, Longchuan, Li, Xiaoqin, Nikolovska-Coleska, Zaneta, McEachern, Donna, Yang, Chao-Yie, Qiu, Su, Yi, Han, Sun, Duxin, Wang, Shaomeng
Publicado em 2011

Targeted Delivery of Paclitaxel to Tumor Cells: Synthesis and In Vitro Evaluation

Por Ndungu, John M., Lu, Yang J., Zhu, Shijun, Yang, Chao, Wang, Xu, Chen, Georgia, Shin, Dong M., Snyder, James P., Shoji, Mamoru, Sun, Aiming
Publicado em 2010

Synthesis and Structure-Activity Relationships of Linear and Conformationally Constrained Peptide Analogs of CIYKYY as Src Tyrosine Kinase Inhibitors

Por Kumar, Anil, Ye, Guofeng, Wang, Yuehao, Lin, Xiaofeng, Sun, Gongqin, Parang, Keykavous
Publicado em 2006

Use of PROTACS as molecular probes of angiogenesis

Por Bargagna-Mohan, Paola, Baek, Sun-Hee, Lee, Hyosung, Kim, Kyungbo, Mohan, Royce
Publicado em 2005

Synthesis and biological evaluation of 3-arylcoumarin derivatives as potential anti-diabetic agents

Por Hu, Yuheng, Wang, Bing, Yang, Jie, Liu, Teng, Sun, Jie, Wang, Xiaojing
Publicado no J Enzyme Inhib Med Chem (2018)

Novel (64)Cu-Radiolabeled Bile Acid Conjugates for Targeted PET Imaging

Por Chong, Hyun-Soon, Chen, Yunwei, Kang, Chi Soo, Sun, Xiang, Wu, Ningjie
Publicado no Bioorg Med Chem Lett (2015)

A new (18)F-labeled BBN-RGD peptide heterodimer with a symmetric linker for prostate cancer imaging

Por Yan, Yongjun, Chen, Kai, Yang, Min, Sun, Xilin, Liu, Shuanglong, Chen, Xiaoyuan
Publicado em 2010

IVSPlat 1.0: an integrated virtual screening platform with a molecular graphical interface

Por Sun, Yin Xue, Huang, Yan Xin, Li, Feng Li, Wang, Hong Yan, Fan, Cong, Bao, Yong Li, Sun, Lu Guo, Ma, Zhi Qiang, Kong, Jun, Li, Yu Xin
Publicado em 2012

Effect of anchoring 4-anilidopiperidines to opioid peptides

Por Petrov, Ravil R., Lee, Yeon Sun, Vardanyan, Ruben S., Liu, Lu, Ma, Shou-wu, Davis, Peg, Lai, Josephine, Porreca, Frank, Vanderah, Todd W., Hruby, Victor J.
Publicado em 2013

Design, synthesis, and biological evaluation of a new class of small molecule peptide mimetics targeting the melanocortin receptors

Por Cain, James P., Mayorov, Alexander V., Cai, Minying, Wang, Hui, Tan, Bahar, Chandler, Kevin, Lee, YeonSun, Petrov, Ravil R., Trivedi, Dev, Hruby, Victor J.
Publicado em 2006

Modification of Amphipathic Non-opioid Dynorphin A Analogues for Rat Brain Bradykinin Receptors

Por Lee, Yeon Sun, Hall, Sara M., Ramos-Colon, Cyf, Remesic, Michael, LeBaron, Lindsay, Nguyen, Ann, Rankin, David, Porreca, Frank, Lai, Josephine, Hruby, Victor J.
Publicado no Bioorg Med Chem Lett (2014)

Non-nucleoside inhibitors of the measles virus RNA-dependent RNA polymerase complex activity: synthesis and in vitro evaluation

Por Sun, Aiming, Chandrakumar, Nizal, Yoon, Jeong-Joong, Plemper, Richard K., Snyder, James P.
Publicado em 2007

A comparative study of trans- and cis-isomers of a bone-seeking agent, DO2A2P

Por Hao, Guiyang, Liu, Wei, Hassan, Gedaa, Öz, Orhan K., Kovacs, Zoltan, Sun, Xiankai
Publicado no Bioorg Med Chem Lett (2014)

Microbeads-Guided Reconstruction of 3D Osteocyte Network during Microfluidic Perfusion Culture

Por Gu, Yexin, Zhang, Wenting, Sun, Qiaoling, Hao, Yi, Zilberberg, Jenny, Lee, Woo Y.
Publicado no J Mater Chem B Mater Biol Med (2015)

A novel model mouth system for evaluation of In Vitro release of nicotine from moist snuff

Por Li, Peng, Zhang, Jie, Sun, Shi-Hao, Xie, Jian-Ping, Zong, Yong-Li
Publicado em 2013

Synthesis and Evaluation of Aryl Quinolines as HIV-1 Integrase Multimerization Inhibitors

Por Jentsch, Nicholas G., Hart, Alison P., Hume, Jared D., Sun, Jian, McNeely, Kaitlin A., Lama, Chiyang, Pigza, Julie A., Donahue, Matthew G., Kessl, Jacques J.
Publicado no ACS Med Chem Lett (2018)

Surface-enhanced Raman spectroscopy investigation on human breast cancer cells

Por Zhu, Jichun, Zhou, Jing, Guo, Jianyu, Cai, Weiying, Liu, Bo, Wang, Zugeng, Sun, Zhenrong
Publicado em 2013