Understanding the structural requirements of 4-anilidopiperidine analogues for biological activities at μ and δ opioid receptors

par Lee, Yeon Sun, Nyberg, Joel, Moye, Sharif, Agnes, Richard S., Davis, Peg, Ma, Shou-wu, Lai, Josephine, Porreca, Frank, Vardanyan, Ruben, Hruby, Victor J.
Publié 2007

Discovery of tripeptide-derived multifunctional ligands possessing delta/mu opioid receptor agonist and neurokinin 1 receptor antagonist activities

par Nair, Padma, Yamamoto, Takashi, Cowell, Scott, Kulkarni, Vinod, Moye, Sharif, Navratilova, Edita, Davis, Peg, Ma, Shou-Wu, Vanderah, Todd W., Lai, Josephine, Porreca, Frank, Hruby, Victor J.
Publié dans Bioorg Med Chem Lett (2015)

Design, Synthesis, and Biological Evaluation of Novel Bifunctional C-Terminal-Modified Peptides for δ/μ Opioid Receptor Agonists and Neurokinin-1 Receptor Antagonists

par Yamamoto, Takashi, Nair, Padma, Davis, Peg, Ma, Shou-wu, Navratilova, Edita, Moye, Sharif, Tumati, Suneeta, Lai, Josephine, Vanderah, Todd W., Yamamura, Henry I., Porreca, Frank, Hruby, Victor J.
Publié 2007

The Importance of Micelle-Bound States for the Bioactivities of Bifunctional Peptide Derivatives for δ/μ Opioid Receptor Agonists and Neurokinin 1 Receptor Antagonists

par Yamamoto, Takashi, Nair, Padma, Jacobsen, Neil E., Davis, Peg, Ma, Shou-wu, Navratilova, Edita, Moye, Sharif, Lai, Josephine, Yamamura, Henry I., Vanderah, Todd W., Porreca, Frank, Hruby, Victor J.
Publié 2008

Novel Bifunctional Peptides as Opioid Agonists and NK-1 Antagonists

par Nair, Padma, Yamamoto, Takashi, Kulkarni, Vinod, Moye, Sharif, Navratilova, Edita, Davis, Peg, Largent, Tally, Ma, Shou-wu, Yamamura, Henry I., Vanderah, Todd, Lai, Josephine, Porreca, Frank, Hruby, Victor. J.
Publié dans Adv Exp Med Biol (2009)

Truncation of the peptide sequence in bifunctional ligands with mu and delta opioid receptor agonist and neurokinin 1 receptor antagonist activities

par Nair, Padma, Yamamoto, Takashi, Largent-Milnes, Tally M., Cowell, Scott, Kulkarni, Vinod, Moye, Sharif, Navratilova, Edita, Davis, Peg, Ma, Shou-Wu, Vanderah, Todd W., Lai, Josephine, Porreca, Frank, Hruby, Victor J.
Publié 2013

A Structure–Activity Relationship Study and Combinatorial Synthetic Approach of C-Terminal Modified Bifunctional Peptides That Are δ/μ Opioid Receptor Agonists and Neurokinin 1 Rec...

par Yamamoto, Takashi, Nair, Padma, Vagner, Josef, Largent-Milnes, Tally, Davis, Peg, Ma, Shou-wu, Navratilova, Edita, Moye, Sharif, Tumati, Suneeta, Lai, Josephine, Yamamura, Henry I., Vanderah, Todd W., Porreca, Frank, Hruby, Victor J.
Publié 2008