SAR Studies on Aromatic Acylhydrazone-Based Inhibitors of Fungal Sphingolipid Synthesis as Next-Generation Antifungal Agents

Por Haranahalli, Krupanandan, Lazzarini, Cristina, Sun, Yi, Zambito, Julia, Pathiranage, Senuri, McCarthy, J. Brian, Mallamo, John, Del Poeta, Maurizio, Ojima, Iwao
Publicado no J Med Chem (2019)

Deglycase-activity oriented screening to identify DJ-1 inhibitors

Por Maksimovic, Igor, Finkin-Groner, Efrat, Fukase, Yoshiyuki, Zheng, Qingfei, Sun, Shan, Michino, Mayako, Huggins, David J., Myers, Robert W., David, Yael
Publicado no RSC Med Chem (2021)

Synthesis of 5-isoxazol-5-yl-2′-deoxyuridines exhibiting antiviral activity against HSV and several RNA viruses

Por Lee, Yoon-Suk, Park, Sun Min, Kim, Byeang Hyean
Publicado no Bioorg Med Chem Lett (2009)

Quaternized chitosans bind onto preexisting biofilms and eradicate pre-attached microorganisms

Por Jiang, Fuguang, Deng, Ying, Yeh, Chih-Ko, Sun, Yuyu
Publicado no J Mater Chem B Mater Biol Med (2014)

DNA cleavage induced by antitumor antibiotic leinamycin and its biological consequences

Por Viswesh, Velliyur, Hays, Allison M., Gates, Kent, Sun, Daekyu
Publicado em 2012

Development of novel enkephalin analogues which have enhanced opioid activities at both μ and δ opioid receptors

Por Lee, Yeon Sun, Petrov, Ravil, Park, Chad K., Ma, Shou-wu, Davis, Peg, Lai, Josephine, Porreca, Frank, Vardanyan, Ruben, Hruby, Victor J.
Publicado em 2007

Thioxo-dihydroquinazolin-one Compounds as Novel Inhibitors of Myeloperoxidase

Por Li, Yang, Ganesh, Thota, Diebold, Becky A., Zhu, Yerun, McCoy, James W., Smith, Susan M. E., Sun, Aiming, Lambeth, J. David
Publicado no ACS Med Chem Lett (2015)

Cyclic non-opioid dynorphin A analogues for the bradykinin receptors

Por Lee, Yeon Sun, Remesic, Michael, Ramos-Colon, Cyf, Hall, Sara M., Kuzmin, Alexander, Rankin, David, Porreca, Frank, Lai, Josephine, Hruby, Victor J.
Publicado no Bioorg Med Chem Lett (2016)

Potent and Selective Double-Headed Thiophene-2-carboximidamide Inhibitors of Neuronal Nitric Oxide Synthase for the Treatment of Melanoma

Por Huang, He, Li, Huiying, Yang, Sun, Chreifi, Georges, Martásek, Pavel, Roman, Linda J., Meyskens, Frank L., Poulos, Thomas L., Silverman, Richard B.
Publicado em 2014

Optimization of Dipeptidic Inhibitors of Cathepsin L for Improved Toxoplasma gondii Selectivity and CNS Permeability

Por Zwicker, Jeffery D., Diaz, Nicolas A., Guerra, Alfredo J., Kirchhoff, Paul D., Wen, Bo, Sun, Duxin, Carruthers, Vern B., Larsen, Scott D.
Publicado no Bioorg Med Chem Lett (2018)

Toward Orally Absorbed Prodrugs of the Antibiotic Aztreonam. Design of Novel Prodrugs of Sulfate Containing Drugs. Part 2

Por Gordon, Eric M., Duncton, Matthew A. J., Wang, Brian J., Qi, Longwu, Fan, Dazhong, Li, Xianfeng, Ni, Zhi-Jie, Ding, Pingyu, Grygorash, Ruslan, Low, Eddy, Yu, Guijun, Sun, Jiawei
Publicado no ACS Med Chem Lett (2020)

A study of inhibitors of d-glycero-β-d-manno-heptose-1-phosphate adenylyltransferase from Burkholderia pseudomallei as a potential antibiotic target

Por Kim, Suwon, Jo, Seri, Kim, Mi-Sun, Shin, Dong Hae
Publicado no J Enzyme Inhib Med Chem (2021)

Derivatization of (±) dihydrotetrabenazine for copper-64 labeling towards long-lived radiotracers for PET imaging of the vesicular monoamine transporter 2

Por Kumar, Amit, Lo, Su-Tang, Öz, Orhan K., Sun, Xiankai
Publicado no Bioorg Med Chem Lett (2014)

Design, radiosynthesis, and evaluation of radiotracers for positron emission tomography imaging of stearoyl-CoA desaturase-1

Por Silvers, William C., Cai, Hancheng, Öz, Orhan K., Sun, Xiankai
Publicado no Bioorg Med Chem Lett (2015)

Synthesis and biological evaluation of 3-arylbenzofuranone derivatives as potential anti-Alzheimer’s disease agents

Por Yang, Jie, Yun, Yinling, Miao, Yuhang, Sun, Jie, Wang, Xiaojing
Publicado no J Enzyme Inhib Med Chem (2020)

Inhibition of African swine fever virus protease by myricetin and myricitrin

Por Jo, Seri, Kim, Suwon, Shin, Dong Hae, Kim, Mi-Sun
Publicado no J Enzyme Inhib Med Chem (2020)

Synthesis and anti-rheumatoid arthritis activities of 3-(4-aminophenyl)-coumarin derivatives

Por Miao, Yuhang, Yang, Jie, Yun, Yinling, Sun, Jie, Wang, Xiaojing
Publicado no J Enzyme Inhib Med Chem (2021)

An overview on natural farnesyltransferase inhibitors for efficient cancer therapy

Por Dai, Xiaohan, Sun, Yingni, Zhang, Ting, Ming, Yongfei, Hongwei, Gao
Publicado no J Enzyme Inhib Med Chem (2020)

A study of Rose Bengal against a 2-keto-3-deoxy-d-manno-octulosonate cytidylyltransferase as an antibiotic candidate

Por Kim, Suwon, Jo, Seri, Kim, Mi-Sun, Shin, Dong Hae
Publicado no J Enzyme Inhib Med Chem (2020)

Cobalt metal-organic framework modified carbon cloth/paper hybrid electrochemical button-sensor for nonenzymatic glucose diagnostics

Por Wei, Xiaofeng, Guo, Jialei, Lian, Huiting, Sun, Xiangying, Liu, Bin
Publicado no Sens Actuators B Chem (2021)