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Synthesis of 5-isoxazol-5-yl-2′-deoxyuridines exhibiting antiviral activity against HSV and several RNA viruses

This paper describes a simple method for synthesizing a small library of 5-isoxazol-5-yl-2′-deoxyuridines from 5-iodo-2′-deoxyuridine. Nitrile oxides were generated in situ from oximes using a commercial bleaching agent; their cycloaddition with 5-ethynyl-2′-deoxyuridine yielded isoxazoles possessin...

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Bibliographic Details
Published in:Bioorg Med Chem Lett
Main Authors: Lee, Yoon-Suk, Park, Sun Min, Kim, Byeang Hyean
Format: Artigo
Language:Inglês
Published: Published by Elsevier Ltd. 2009
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC7126966/
https://ncbi.nlm.nih.gov/pubmed/19147352
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2008.12.103
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