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In Vitro–In Vivo Inaccuracy: The CYP3A4 Anomaly

When predicting hepatic clearance using in vitro to in vivo extrapolation (IVIVE), microsomes or hepatocytes are commonly used. Here, we examine intrinsic clearance values and IVIVE results in human hepatocytes and microsomes for compounds metabolized by a variety of enzymes. The great majority of C...

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Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:Drug Metab Dispos
Prif Awduron: Bowman, Christine M., Benet, Leslie Z.
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: The American Society for Pharmacology and Experimental Therapeutics 2019
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC7042718/
https://ncbi.nlm.nih.gov/pubmed/31551322
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.119.088427
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