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The Presence of a Transporter-Induced Protein Binding Shift: A New Explanation for Protein-Facilitated Uptake and Improvement for In Vitro-In Vivo Extrapolation

Accurately predicting hepatic clearance is an integral part of the drug-development process, and yet current in vitro to in vivo (IVIVE) extrapolation methods yield poor predictions, particularly for highly protein-bound transporter substrates. Explanations for error include inaccuracies in protein-...

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Detalhes bibliográficos
Publicado no:Drug Metab Dispos
Main Authors: Bowman, Christine M., Okochi, Hideaki, Benet, Leslie Z.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6413769/
https://ncbi.nlm.nih.gov/pubmed/30674616
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.118.085779
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