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Investigating the Theoretical Basis for In Vitro-In Vivo Extrapolation (IVIVE) in Predicting Drug Metabolic Clearance and Proposing Future Experimental Pathways
INTRODUCTION: Extensive studies have been conducted to predict in vivo metabolic clearance from in vitro human liver metabolism parameters (i.e., in vitro-in vivo-extrapolation; IVIVE) with little success. METHODS: Here, deriving IVIVE from first principles, we show that the product of fraction unbo...
Tallennettuna:
| Julkaisussa: | AAPS J |
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| Päätekijät: | , |
| Aineistotyyppi: | Artigo |
| Kieli: | Inglês |
| Julkaistu: |
2020
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| Aiheet: | |
| Linkit: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7515557/ https://ncbi.nlm.nih.gov/pubmed/32914238 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-020-00501-9 |
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