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The Pharmacology of Cyclopropyl-Methoxycarbonyl Metomidate: A Comparison with Propofol

BACKGROUND: Cyclopropyl-methoxycarbonyl metomidate (CPMM) is a “soft” etomidate analogue currently being developed as a propofol alternative for anesthetic induction and maintenance. METHODS: We compared the potencies of CPMM and propofol by assessing their abilities to directly activate α(1)(L264T)...

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Pubblicato in:Anesth Analg
Autori principali: Ge, Rile, Pejo, Ervin, Gallin, Hilary, Jeffrey, Spencer, Cotten, Joseph F., Raines, Douglas E.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6310170/
https://ncbi.nlm.nih.gov/pubmed/24557104
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1213/ANE.0000000000000069
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