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Autoinhibition in Ras effectors Raf, PI3Kα, and RASSF5: a comprehensive review underscoring the challenges in pharmacological intervention

Autoinhibition is an effective mechanism that guards proteins against spurious activation. Despite its ubiquity, the distinct organizations of the autoinhibited states and their release mechanisms differ. Signaling is most responsive to the cell environment only if a small shift in the equilibrium i...

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Dettagli Bibliografici
Pubblicato in:Biophys Rev
Autori principali: Nussinov, Ruth, Zhang, Mingzhen, Tsai, Chung-Jung, Liao, Tsung-Jen, Fushman, David, Jang, Hyunbum
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer Berlin Heidelberg 2018
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6233353/
https://ncbi.nlm.nih.gov/pubmed/30269291
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s12551-018-0461-0
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