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Development of novel fluorescent histamine H(1)-receptor antagonists to study ligand-binding kinetics in living cells

The histamine H(1)-receptor (H(1)R) is an important mediator of allergy and inflammation. H(1)R antagonists have particular clinical utility in allergic rhinitis and urticaria. Here we have developed six novel fluorescent probes for this receptor that are very effective for high resolution confocal...

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Détails bibliographiques
Publié dans:Sci Rep
Auteurs principaux: Stoddart, Leigh A., Vernall, Andrea J., Bouzo-Lorenzo, Monica, Bosma, Reggie, Kooistra, Albert J., de Graaf, Chris, Vischer, Henry F., Leurs, Rob, Briddon, Stephen J., Kellam, Barrie, Hill, Stephen J.
Format: Artigo
Langue:Inglês
Publié: Nature Publishing Group UK 2018
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5785503/
https://ncbi.nlm.nih.gov/pubmed/29371669
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-018-19714-2
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