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Subtype-Specific Agonists for NMDA Receptor Glycine Binding Sites
A series of analogues based on serine as lead structure were designed, and their agonist activities were evaluated at recombinant NMDA receptor subtypes (GluN1/2A–D) using two-electrode voltage-clamp (TEVC) electrophysiology. Pronounced variation in subunit-selectivity, potency, and agonist efficacy...
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| Yayımlandı: | ACS Chem Neurosci |
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| Asıl Yazarlar: | , , , , , , , , , , |
| Materyal Türü: | Artigo |
| Dil: | Inglês |
| Baskı/Yayın Bilgisi: |
2017
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| Konular: | |
| Online Erişim: | https://ncbi.nlm.nih.gov/pmc/articles/PMC5559341/ https://ncbi.nlm.nih.gov/pubmed/28514141 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.7b00117 |
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