Загрузка...
Subtype-Specific Agonists for NMDA Receptor Glycine Binding Sites
A series of analogues based on serine as lead structure were designed, and their agonist activities were evaluated at recombinant NMDA receptor subtypes (GluN1/2A–D) using two-electrode voltage-clamp (TEVC) electrophysiology. Pronounced variation in subunit-selectivity, potency, and agonist efficacy...
Сохранить в:
| Опубликовано в: : | ACS Chem Neurosci |
|---|---|
| Главные авторы: | , , , , , , , , , , |
| Формат: | Artigo |
| Язык: | Inglês |
| Опубликовано: |
2017
|
| Предметы: | |
| Online-ссылка: | https://ncbi.nlm.nih.gov/pmc/articles/PMC5559341/ https://ncbi.nlm.nih.gov/pubmed/28514141 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.7b00117 |
| Метки: |
Добавить метку
Нет меток, Требуется 1-ая метка записи!
|