Rational modulation of the induced-fit conformational change for slow-onset inhibition in M. tuberculosis InhA

Eitemau Tebyg

• A Structural and Energetic Model for the Slow-Onset Inhibition of the Mycobacterium tuberculosis Enoyl-ACP Reductase InhA
  gan: Li, Huei-Jiun, et al.
  Cyhoeddwyd: (2014)
• Time-dependent diaryl ether inhibitors of InhA: SAR studies of enzyme inhibition, antibacterial activity, and in vivo efficacy
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  Cyhoeddwyd: (2014)
• Formulation Studies of InhA inhibitors and Combination therapy to improve efficacy against Mycobacterium tuberculosis
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  Cyhoeddwyd: (2016)
• Slow-Onset Inhibition of Mycobacterium tuberculosis InhA: Revealing Molecular Determinants of Residence Time by MD Simulations
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  Cyhoeddwyd: (2015)
• A Slow, Tight Binding Inhibitor of InhA, the Enoyl-Acyl Carrier Protein Reductase from Mycobacterium tuberculosis
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  Cyhoeddwyd: (2010)