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Slow-Onset Inhibition of Mycobacterium tuberculosis InhA: Revealing Molecular Determinants of Residence Time by MD Simulations

An important kinetic parameter for drug efficacy is the residence time of a compound at a drug target, which is related to the dissociation rate constant k(off). For the essential antimycobacterial target InhA, this parameter is most likely governed by the ordering of the flexible substrate binding...

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Xehetasun bibliografikoak
Argitaratua izan da:PLoS One
Egile Nagusiak: Merget, Benjamin, Sotriffer, Christoph A.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Public Library of Science 2015
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4440617/
https://ncbi.nlm.nih.gov/pubmed/25996598
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0127009
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