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A Potent, Selective and Cell-active Inhibitor of Human Type I Protein Arginine Methyltransferases

Protein arginine methyltransferases (PRMTs) play a crucial role in a variety of biological processes. Overexpression of PRMTs has been implicated in various human diseases including cancer. Consequently, selective small-molecule inhibitors of PRMTs have been pursued by both academia and pharmaceutic...

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Bibliografski detalji
Izdano u:ACS Chem Biol
Glavni autori: Eram, Mohammad S., Shen, Yudao, Szewczyk, Magdalena, Wu, Hong, Senisterra, Guillermo, Li, Fengling, Butler, Kyle V., Kaniskan, H. Ümit, Speed, Brandon A., dela Seña, Carlo, Dong, Aiping, Zeng, Hong, Schapira, Matthieu, Brown, Peter J., Arrowsmith, Cheryl H., Barsyte-Lovejoy, Dalia, Liu, Jing, Vedadi, Masoud, Jin, Jian
Format: Artigo
Jezik:Inglês
Izdano: 2015
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4798913/
https://ncbi.nlm.nih.gov/pubmed/26598975
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.5b00839
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