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Mechanistic Insights into Allosteric Structure-Function Relationships at the M(1) Muscarinic Acetylcholine Receptor

Benzylquinolone carboxylic acid (BQCA) is the first highly selective positive allosteric modulator (PAM) for the M(1) muscarinic acetylcholine receptor (mAChR), but it possesses low affinity for the allosteric site on the receptor. More recent drug discovery efforts identified 3-((1S,2S)-2-hydroxycy...

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Détails bibliographiques
Publié dans:J Biol Chem
Auteurs principaux: Abdul-Ridha, Alaa, Lane, J. Robert, Mistry, Shailesh N., López, Laura, Sexton, Patrick M., Scammells, Peter J., Christopoulos, Arthur, Canals, Meritxell
Format: Artigo
Langue:Inglês
Publié: American Society for Biochemistry and Molecular Biology 2014
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Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4246120/
https://ncbi.nlm.nih.gov/pubmed/25326383
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M114.604967
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