Structure–Activity Relationships of Quinoxaline-Based 5-HT(3)A and 5-HT(3)AB Receptor-Selective Ligands

Until recently, discriminating between homomeric 5-HT(3)A and heteromeric 5-HT(3)AB receptors was only possible with ligands that bind in the receptor pore. This study describes the first series of ligands that can discriminate between these receptor types at the level of the orthosteric binding sit...

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Hlavní autoři: Thompson, Andrew J, Verheij, Mark H P, van Muijlwijk-Koezen, Jacqueline E, Lummis, Sarah C R, Leurs, Rob, de Esch, Iwan J P
Médium: Artigo
Jazyk:Inglês
Vydáno: WILEY-VCH Verlag 2013
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On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4063337/
https://ncbi.nlm.nih.gov/pubmed/23640722
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201300032
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