Lataa...

Repurposing human Aurora kinase inhibitors as leads for anti-protozoan drug discovery

Hesperadin, an established human Aurora B inhibitor, was tested against cultures of Trypanosoma brucei, Leishmania major, and Plasmodium falciparum, and was identified to be a potent proliferation inhibitor. A series of analogs was designed and tested to establish the initial structure-activity rela...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Päätekijät: Patel, Gautam, Roncal, Norma E., Lee, Patricia J., Leed, Susan E., Erath, Jessey, Rodriguez, Ana, Sciotti, Richard J., Pollastri, Michael P.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2014
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC4045489/
https://ncbi.nlm.nih.gov/pubmed/24910766
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C4MD00045E
Tagit: Lisää tagi
Ei tageja, Lisää ensimmäinen tagi!