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Biological Effects of the Pim Kinase Inhibitor, SGI-1776, in Multiple Myeloma

Pim kinases are constitutively active serine/threonine/tyrosine kinases that are overexpressed in hematological malignancies such as multiple myeloma. Pim kinase substrates are involved in transcription, protein translation, cell proliferation, and apoptosis. SGI-1776 is a potent Pim kinase inhibito...

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Bibliografske podrobnosti
Main Authors: Cervantes-Gomez, Fabiola, Chen, Lisa S., Orlowski, Robert Z., Gandhi, Varsha
Format: Artigo
Jezik:Inglês
Izdano: 2013
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC3951475/
https://ncbi.nlm.nih.gov/pubmed/23988451
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.clml.2013.05.019
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